BDBM50030727 4''-[3-Butyl-5-oxo-1-(2-trifluoromethyl-phenyl)-1,5-dihydro-[1,2,4]triazol-4-ylmethyl]-biphenyl-2-sulfonic acid benzoylamide::CHEMBL279629::CHEMBL97539::L-159,913::L-159913
SMILES CCCCc1nn(-c2ccccc2C(F)(F)F)c(=O)n1Cc1ccc(cc1)-c1ccccc1S(=O)(=O)NC(=O)c1ccccc1
InChI Key InChIKey=JVOGASLNIGJLLS-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 20 hits for monomerid = 50030727
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
The M. S. University Of Baroda
Curated by ChEMBL
The M. S. University Of Baroda
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:In vitro binding affinity of the compound towards Angiotensin II receptor, type 2 to displace 125I[Sar,Ile] from rat brain tissue preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.330nMAssay Description:In vitro binding affinity of the compound towards Angiotensin II receptor, type 1 to displace 125I[Sar,Ile] from rat adrenal tissue preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:In vitro inhibitory activity against angiotensin II rabbit aorta AT1 receptor using radioligand [125I]-Sar Ile-AIIMore data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 1 in rabbit aorta membrane preparations.More data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Antagonist activity at AT1 receptor in rabbit aorta membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in rat midbrain membrane preparations.More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:In vitro binding affinity against angiotensin II (AT2) receptor to competitively block the specific binding of [125I]- [Sar1,Ile8] AII to a rat mid b...More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:In vitro inhibitory activity against angiotensin II rat midbrain AT2 receptor using radioligand [125I]-Sar Ile-AIIMore data for this Ligand-Target Pair
Affinity DataIC50: 0.310nMAssay Description:In vitro binding affinity of the compound towards Angiotensin II receptor, type 1 to displace 125I[Sar,Ile] from rat brain tissue preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.550nMAssay Description:In vitro binding affinity of the compound towards angiotensin-1 receptor to displace 125I[Sar,Ile] from rabbit brain tissue preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:In vitro binding affinity of the compound towards Angiotensin II receptor, type 2 to displace 125I[Sar,Ile] from rat adrenal tissue preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Inhibitory activity at Angiotensin II type 2 receptor.More data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Displacement of 125I[Sar,Ile] from rabbit aorta membrane Angiotensin II receptor type 1More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:In vitro binding affinity of the compound towards angiotensin-1 receptor to displace 125I[Sar,Ile] from rabbit adrenal tissue preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.550nMAssay Description:In vitro binding affinity of the compound towards angiotensin-1 receptor to displace 125I[Sar,Ile] from rabbit brain tissue preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Tested for in vitro binding affinity against angiotensin I (AT1) receptor to competitively block the specific binding of [125I]- [Sar1,Ile8] AII to a...More data for this Ligand-Target Pair