BDBM120262 EDROPHONIUM BROMIDE::EDROPHONIUM CHLORIDE::Edrophonium::Edrophonium Chloride, 3::cid_8307
SMILES CC[N+](C)(C)c1cccc(O)c1
InChI Key InChIKey=VWLHWLSRQJQWRG-UHFFFAOYSA-O
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 27 hits for monomerid = 120262
Affinity DataKi: 1.60nMAssay Description:Inhibition constant determined against Acetylcholinesterase (AChE) receptor.Checked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity against Acetylcholinesterase of purified calf forebrain (CFB)More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity against Acetylcholinesterase of human RBCMore data for this Ligand-Target Pair
Affinity DataKi: 250nM ΔG°: -9.00kcal/molepH: 7.0 T: 2°CAssay Description:Assays were conducted at 25 C in 20 mM sodium phosphate buffer (pH 7.0) and 0.01% bovine serum albumin unless otherwise noted. AChE concentrations we...More data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Binding affinity against Acetylcholinesterase of purified Octopus brain (OB)More data for this Ligand-Target Pair
Affinity DataKi: 790nMAssay Description:Dissociation constant for enzyme-inhibitor complex of human recombinant AChE by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Inhibition of human erythrocytes recombinant AChE assessed as dissociation constant for enzyme-inhibitor complexMore data for this Ligand-Target Pair
Affinity DataKi: 1.01E+3nMAssay Description:Inhibition constant using AChE or BuChE.More data for this Ligand-Target Pair
Affinity DataKi: 4.80E+3nMAssay Description:Inhibition of human erythrocytes recombinant AChE assessed as dissociation constant for enzyme-inhibitor-substrate complexMore data for this Ligand-Target Pair
Affinity DataKi: 4.80E+3nMAssay Description:Dissociation constant for enzyme-inhibitor-substrate complex of human recombinant AChE by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 4.80E+3nMAssay Description:Competitive inhibition of human recombinant AChE using ATChCl as substrate by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 1.98E+5nMAssay Description:Inhibition constant using AChE or BuChE.More data for this Ligand-Target Pair
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
National Chung-Hsing University
Curated by ChEMBL
National Chung-Hsing University
Curated by ChEMBL
Affinity DataKi: 3.40E+5nMAssay Description:Compound was evaluated for irreversible inhibition of Horse serum ButyrylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.36E+3nMAssay Description:Inhibition of bovine AChEMore data for this Ligand-Target Pair
Affinity DataIC50: 780nMAssay Description:Inhibitory activity against AcetylcholinesteraseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.37E+6nMAssay Description:Inhibition of human plasmatic BChE by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.37E+6nMAssay Description:Inhibition of human plasmatic BChE by modified Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human erythrocyte recombinant AChE by modified Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 5.17E+3nMAssay Description:Inhibition of human recombinant AChE by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.96E+3nMAssay Description:In vitro inhibitory activity against human recombinant AChEMore data for this Ligand-Target Pair
Affinity DataIC50: 780nMAssay Description:Inhibition acetylcholinesterase (AChE) enzyme.More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of Acetylcholinesterase activity of calf forebrainMore data for this Ligand-Target Pair
Affinity DataIC50: 5.17E+3nMAssay Description:Inhibition of human recombinant AChE after 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.37E+6nMAssay Description:Inhibition of human plasmatic BChE after 5 mins by Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of Acetylcholinesterase activity from octopus brainMore data for this Ligand-Target Pair
Affinity DataIC50: >5.00E+4nMAssay Description:The HTS assay to identify Inhibitors of West Nile Virus (WNV) NS2bNS3 Proteinase was proposed by Dr Alex Strongin of the Burnham Institute XO1-MH0776...More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of Acetylcholinesterase from human red blood cellsMore data for this Ligand-Target Pair