BDBM50094687 1-(8-Butyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-methoxy-phenyl)-urea::1-(8-butyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-yl)-3-(4-methoxyphenyl)urea::CHEMBL330286
SMILES CCCCn1cc2c(n1)nc(NC(=O)Nc1ccc(OC)cc1)n1nc(nc21)-c1ccco1
InChI Key InChIKey=XMCVJFCDPDUAPT-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 19 hits for monomerid = 50094687
Affinity DataIC50: 4.10nMAssay Description:Inhibition of cAMP accumulation in CHO cells expressing human adenosine A3 receptor; range 2.9-6.0More data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells; range 0.27-0.34More data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Displacement of [3H]MRE3008-F20 from human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Binding affinity for human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Displacement of [3H]MRE3008-F20 from human Adenosine A3 receptor expressed in HEK cells; range 0.27-0.34More data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Displacement of [3H]-SCH- 58261 from human adenosine A2A receptor expressed in CHO cells; range 65-92More data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Displacement of [3H]SCH-58261 from human Adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 80nMAssay Description:Displacement of [3H]SCH-58261 from human Adenosine A2A receptor expressed in HEK293 cells; range 65-92More data for this Ligand-Target Pair
Affinity DataKi: 296nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells; range 269-326More data for this Ligand-Target Pair
Affinity DataKi: 296nMAssay Description:Displacement of [3H]-DPCPX from human Adenosine A1 receptor expressed in CHO cells; range 269-326More data for this Ligand-Target Pair
Affinity DataKi: 296nMAssay Description:Displacement of [3H]DPCPX from human Adenosine A1 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 303nMAssay Description:Displacement of [3H]DPCPX from human Adenosine A2B receptor expressed in HEK293 cells; range 262-352More data for this Ligand-Target Pair
Affinity DataKi: 303nMAssay Description:Displacement of [3H]DPCPX from human Adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 303nMAssay Description:Displacement of [3H]DPCPX from Adenosine A2b receptor expressed in CHO cells; range 260-352More data for this Ligand-Target Pair
Affinity DataKi: 324nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair