BDBM50177300 CHEMBL379886::N-(2-(2-(dimethylamino)ethylamino)-4-methylquinolin-6-yl)-2-(4-(trifluoromethoxy)phenoxy)acetamide

SMILES CN(C)CCNc1cc(C)c2cc(NC(=O)COc3ccc(OC(F)(F)F)cc3)ccc2n1

InChI Key InChIKey=LGMXSRRDGDVUCC-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50177300   

TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50177300(CHEMBL379886 | N-(2-(2-(dimethylamino)ethylamino)-...)
Affinity DataIC50:  5.30nMAssay Description:Displacement of [125I]MCH from human MCH1 receptor expressed in CHO cell by WC assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50177300(CHEMBL379886 | N-(2-(2-(dimethylamino)ethylamino)-...)
Affinity DataIC50:  18nMAssay Description:Inhibition of human MCH1 receptor by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed