BDBM50224401 8-(4-chlorophenyl)-1h-pyrazolo[3'',4'':4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-7(8H)-one::CHEMBL238263

SMILES Clc1ccc(cc1)-n1cnc2c(sc3ncc4c[nH]nc4c23)c1=O

InChI Key InChIKey=LKBNBRKQCADHSO-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50224401   

TargetMetabotropic glutamate receptor 1(Human)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50224401(8-(4-chlorophenyl)-1h-pyrazolo[3'',4'':4',5']pyrid...)
Affinity DataIC50:  38nMAssay Description:Antagonist activity at human mGluR1a expressed in CHO cells assessed by measuring intracellular calcium by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed