BDBM50345261 CHEMBL1782532::cis-5-bromo-7-(4-hydroxycyclohexylamino)benzofuran-2-carboxylic acid

SMILES O[C@H]1CC[C@H](CC1)Nc1cc(Br)cc2cc(oc12)C(O)=O

InChI Key InChIKey=IQNDSBJQOZFMDJ-PHIMTYICSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50345261   

TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50345261(CHEMBL1782532 | cis-5-bromo-7-(4-hydroxycyclohexyl...)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of human Pim2 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 90 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Genzyme

Curated by ChEMBL
LigandPNGBDBM50345261(CHEMBL1782532 | cis-5-bromo-7-(4-hydroxycyclohexyl...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human Pim1 using 5-FAM-RSRHSSYPAGT-CONH2 as substrate after 45 mins by off-chip mobility shift methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed