BDBM50395176 CHEMBL2163952

SMILES CC12CC3CC(C)(C1)CC(C3)(C2)NC(=O)c1cn2C(COc3cccc(c23)c1=O)c1ccccc1

InChI Key InChIKey=ADAWJIUDJGXERN-UHFFFAOYSA-N

Data  4 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50395176   

TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50395176(CHEMBL2163952)
Affinity DataKi:  3.45nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in CHO cell membranes incubated for 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50395176(CHEMBL2163952)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]CP-55940 from CB2 receptor in Sprague-Dawley rat spleen by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50395176(CHEMBL2163952)
Affinity DataKi:  460nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB1 receptor expressed in CHO cell membranes incubated for 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50395176(CHEMBL2163952)
Affinity DataKi:  545nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in Sprague-Dawley rat brain by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed