BDBM50395751 CHEMBL2164507

SMILES CCN1CCC(CC(=O)NC2(C(=O)Nc3cc(Cl)cc(Cl)c23)c2ccc(Cl)c(Cl)c2)CC1

InChI Key InChIKey=RYVLJWQSUMPPDS-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50395751   

TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395751(CHEMBL2164507)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]-ghrelin from human GHSR1 expressed in CHO-CREluc cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395751(CHEMBL2164507)
Affinity DataIC50:  1nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed