BDBM50402487 CHEMBL2204054

SMILES O=c1[nH]c([C@@H]2CC[C@@H](CC2)c2ccccc2)c(Cc2nccs2)c(=O)[nH]1

InChI Key InChIKey=BQKFLGKVHUYRPC-GASCZTMLSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50402487   

TargetGlucocorticoid receptor(Homo sapiens (Human))
Corcept Therapeutics

Curated by ChEMBL
LigandPNGBDBM50402487(CHEMBL2204054)
Affinity DataKi:  139nMAssay Description:Displacement of [3H]dexamethasone from human recombinant glucocorticoid receptor expressed in baculovirus after 18 hrs by scintillation counting anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Corcept Therapeutics

Curated by ChEMBL
LigandPNGBDBM50402487(CHEMBL2204054)
Affinity DataKi: >300nMAssay Description:Antagonist activity at glucocorticoid receptor in human SW1353 cells assessed as inhibition of dexamethasone-induced luciferase expression after 16 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed