BDBM50415388 CHEMBL604524

SMILES CCCc1ccc(cc1)N(C)C(=O)c1c(C)onc1-c1ccccc1Cl

InChI Key InChIKey=CHDRRISOFKAHLC-UHFFFAOYSA-N

Data  1 EC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50415388   

TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
GlaxoSmithKline

Curated by ChEMBL
LigandPNGBDBM50415388(CHEMBL604524)
Show SMILES CCCc1ccc(cc1)N(C)C(=O)c1c(C)onc1-c1ccccc1Cl
Show InChI InChI=1S/C21H21ClN2O2/c1-4-7-15-10-12-16(13-11-15)24(3)21(25)19-14(2)26-23-20(19)17-8-5-6-9-18(17)22/h5-6,8-13H,4,7H2,1-3H3
Affinity DataEC50:  6.31E+3nMAssay Description:Agonist activity at human TGR5 receptor expressed in human U2-OS cells assessed as changes in response to cAMP level by MRE/CRE-driven luciferase rep...More data for this Ligand-Target Pair