BDBM50434295 CHEMBL2386353
SMILES OC(=O)CCc1ccc(cc1F)C#Cc1ccccc1CC#N
InChI Key InChIKey=KIZUBVPJNPVIIN-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 10 hits for monomerid = 50434295
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataKi: 85nMAssay Description:Displacement of 3-(2-Fluoro-4-((2'-methyl-4'-(2-(2-((7-nitrobenzo[c][1,2,5]-oxadiazol-4-yl)amino)ethoxy)ethoxy)-[1,1'-biphenyl]-3-yl)-methoxy)phenyl)...More data for this Ligand-Target Pair
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 5.90nMAssay Description:Agonist activity at FFA1 receptor (unknown origin) expressed in human 132N1 cells measured for 90 secs by Fura-2 AM dye based calcium mobilization as...More data for this Ligand-Target Pair
TargetFree fatty acid receptor 4(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 933nMAssay Description:Agonist activity at C-terminal yellow fluorescent protein-fused human FFA4 receptor transfected in HEK293 cells after 5 mins by BRET assayMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 6.20nMAssay Description:Agonist activity at human FFA1 receptor transfected in human 1321N1 cells by calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataEC50: 148nMAssay Description:Agonist activity at mouse FFA1 receptor transfected in human T-REX-293 cells measured for 74 secs by calcium mobilization assayMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 26nMAssay Description:Agonist activity at C-terminal yellow fluorescent protein-fused human FFA1 receptor transfected in HEK293 cells after 5 mins by BRET assay in presenc...More data for this Ligand-Target Pair
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 23nMAssay Description:Agonist activity at C-terminal yellow fluorescent protein-fused human FFA1 receptor transfected in HEK293 cells after 5 mins by BRET assayMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 6nMAssay Description:Agonist activity at human FFA1 receptor transfected in human 1321N1 cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Agonist activity at human C-terminal eYFP-tagged FFA1 receptor expressed in HEK-293 cells assessed as beta-arrestin2 recruitment incubated for 5 mins...More data for this Ligand-Target Pair
Affinity DataEC50: 324nMAssay Description:Agonist activity at C-terminal yellow fluorescent protein-fused rat FFA1 receptor transfected in HEK293 cells after 5 mins by BRET assayMore data for this Ligand-Target Pair