BDBM50504904 CHEMBL4513684

SMILES NS(=O)(=O)c1cc(C(=O)NCCCC(O)=O)c(SC2CCCCC2)cc1Cl

InChI Key InChIKey=QBFWPSYDISFIKC-UHFFFAOYSA-N

Data  23 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 23 hits for monomerid = 50504904   

TargetCarbonic anhydrase 5A, mitochondrial(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  1.60nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 5a expressed in Escherichia coli expression system assessed as kinetic dissociation constant...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 1(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  3.30E+3nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 1 expressed in Escherichia coli expression system assessed as observed dissociation constant...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 7(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  0.0300nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 7 expressed in Escherichia coli expression system assessed as kinetic dissociation constant ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 12(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  0.400nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 12 expressed in Escherichia coli expression system assessed as observed dissociation constan...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 4(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  130nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 4 expressed in Escherichia coli expression system assessed as observed dissociation constant...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 13(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  1.20nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 13 expressed in Escherichia coli expression system assessed as kinetic dissociation constant...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 13(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  130nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 13 expressed in Escherichia coli expression system assessed as observed dissociation constan...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 9(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  2.20nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 9 expressed in mammalian cell expression system assessed as observed dissociation constant f...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 5A, mitochondrial(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  250nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 5a expressed in Escherichia coli expression system assessed as observed dissociation constan...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 1(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  30nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 1 expressed in Escherichia coli expression system assessed as kinetic dissociation constant ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 2(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  13nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 2 expressed in Escherichia coli expression system assessed as observed dissociation constant...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 5B, mitochondrial(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  0.160nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 5b expressed in Escherichia coli expression system assessed as kinetic dissociation constant...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 2(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  0.0600nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 2 expressed in Escherichia coli expression system assessed as kinetic dissociation constant ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 14(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  0.00700nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 14 expressed in Escherichia coli expression system assessed as kinetic dissociation constant...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 3(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd: >2.00E+5nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 3 expressed in Escherichia coli expression system assessed as kinetic dissociation constant ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 12(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  0.00200nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 12 expressed in Escherichia coli expression system assessed as kinetic dissociation constant...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 5B, mitochondrial(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  33nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 5b expressed in Escherichia coli expression system assessed as observed dissociation constan...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 6(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  2nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 6 expressed in Escherichia coli expression system assessed as kinetic dissociation constant ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 14(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  1.80nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 14 expressed in Escherichia coli expression system assessed as observed dissociation constan...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 4(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  0.350nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 4 expressed in Escherichia coli expression system assessed as kinetic dissociation constant ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 7(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  9.10nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 7 expressed in Escherichia coli expression system assessed as observed dissociation constant...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 6(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  2.20E+3nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 6 expressed in Escherichia coli expression system assessed as observed dissociation constant...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCarbonic anhydrase 9(Human)
Vilnius University

Curated by ChEMBL
LigandPNGBDBM50504904(CHEMBL4513684)
Affinity DataKd:  0.00700nMAssay Description:Binding affinity to recombinant human carbonic anhydrase 9 expressed in mammalian cell expression system assessed as kinetic dissociation constant fl...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed