BDBM50510054 CHEMBL4445209

SMILES Cc1nn(c(C)c1-c1ccc(F)cc1)-c1ccc(CN)cn1

InChI Key InChIKey=POIKSTHXKNCWIR-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50510054   

TargetAcid-sensing ion channel 2(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510054(CHEMBL4445209)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of pH 6.25-stimulated mouse ASIC1a/2a heterodimer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 2(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510054(CHEMBL4445209)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of pH 5.5-stimulated mouse ASIC2a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510054(CHEMBL4445209)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed