BDBM50529442 CHEMBL4458766

SMILES Cn1ncc2cccc(CN3CCN(CC3=O)c3cn[nH]c(=O)c3Cl)c12

InChI Key InChIKey=KLZVSLPAAMLVTO-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50529442   

TargetShort transient receptor potential channel 5(Homo sapiens (Human))
Goldfinch Bio

Curated by ChEMBL
LigandPNGBDBM50529442(CHEMBL4458766)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of rosiglitazone-activated human TRPC5 channel expressed in HEK293 cells assessed as reduction in Ca2+ current measured at +80 mV with hol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed