BDBM50583745 CHEMBL5092736
SMILES CCCCn1c(CC)nc2ccc(nc12)-c1cc(N)nc(N)c1
InChI Key InChIKey=HINVECUKBZWJTC-UHFFFAOYSA-N
Data 3 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50583745
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Servier Research Institute Of Medicinal Chemistry
Curated by ChEMBL
Servier Research Institute Of Medicinal Chemistry
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of DYRK1A (unknown origin) using Ulight-MBP as substrate and ATP as co-substrate incubated for 40 mins and measured after 1 hr by TR-FRET ...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Servier Research Institute Of Medicinal Chemistry
Curated by ChEMBL
Servier Research Institute Of Medicinal Chemistry
Curated by ChEMBL
Affinity DataIC50: 153nMAssay Description:Inhibition of wild type full length DYRK1A (unknown origin) in human U2OS cells assessed as reduction in pSER520 autophosphorylation incubated for 5 ...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Servier Research Institute Of Medicinal Chemistry
Curated by ChEMBL
Servier Research Institute Of Medicinal Chemistry
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK9 (unknown origin) using Ulight-MBP as substrate and ATP as co-substrate incubated for 40 mins and measured after 1 hr by TR-FRET as...More data for this Ligand-Target Pair