BDBM521988 N-[3-[6-(difluoromethoxy)- 3,4-dihydro-2H-1,4- benzothiazin-7-yl]-1-[2- [[(3R)-tetrahydrofuran-3- yl]amino]ethyl]pyrazol-4- yl]pyrazolo[1,5-a]pyrimidine- 3-carboxamide::US11155557, Example 78
SMILES FC(F)Oc1cc2NCCSc2cc1-c1nn(CCN[C@@H]2CCOC2)cc1NC(=O)c1cnn2cccnc12
InChI Key InChIKey=BLVCWVSYQABHSB-OAHLLOKOSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 521988
Affinity DataKi: 0.100nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:The activity of the isolated recombinant JAK1 and JAK2 kinase domain was measured by monitoring phosphorylation of a peptide derived from JAK3 (Val-A...More data for this Ligand-Target Pair