BDBM86248 CAS_364-98-7::NSC_3019::diazoxide

SMILES CC1=Nc2ccc(Cl)cc2S(=O)(=O)N1

InChI Key InChIKey=GDLBFKVLRPITMI-UHFFFAOYSA-N

Data  2 KI  4 IC50  1 Kd  6 EC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 86248   

LigandPNGBDBM86248(CAS_364-98-7 | NSC_3019 | diazoxide)
Affinity DataEC50:  2.35E+4nMAssay Description:Activation of human recombinant SUR1/Kir6.2 channel expressed in HEK293 cells assessed as increase in ionic current by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed