TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of Brsk2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of Brsk2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of human BRSK2 using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human BRSK2 using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of BRSK2 in the presence of 50uM ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of BRSK2 in the presence of 50uM ATPMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of BRSK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of BRSK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of recombinant human BRSK2 (2 to end residues) using KKLNRTLSFAEPG substrate incubated for 40 mins in presence of [gamma-33ATP] by radiome...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human BRSK2 using [KKLNRTLSFAEPG] as substrateMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of BRSK2 (unknown origin)More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 2.70E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 650nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 4.10E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 3.5nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 650nMAssay Description:Binding affinity to BRSK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 16nMAssay Description:Binding affinity to BRSK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 16nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 650nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 3.5nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 3.5nMAssay Description:Binding constant for full-length BRSK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 650nMAssay Description:Binding constant for full-length BRSK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 92nMAssay Description:Binding affinity to human BRSK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to BRSK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to BRSK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to BRSK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to BRSK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Binding affinity to BRSK2More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 190nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 5.60E+3nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase BRSK2(Homo sapiens (Human))
Vertex Pharmaceuticals
Curated by ChEMBL
Vertex Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for BRSK2 kinase domainMore data for this Ligand-Target Pair