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RF 9

* Please kindly note that our products are not to be used for therapeutic purposes and cannot be sold to patients.

RF 9 is a potent and selective Neuropeptide FF receptor antagonist, with Kis of 58±5 and 75±9 nM for hNPFF1R and hNPFF2R, respectively. It displays selectivity over several related receptors including NPY Y1 GPR10, GPR54, GPR103 and the opioid receptors.

Category

Peptide Inhibitors

Catalog number

BAT-010204

CAS number

876310-60-0

Molecular Formula

C26H38N6O3

Molecular Weight

482.62

Specification
Reference Reading

IUPAC Name

N-[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]adamantane-1-carboxamide

Synonyms

2-Adamantanecarbonyl-Arg-Phe-NH2

Purity

≥96%

Density

1.42±0.1 g/cm3(Predicted)

Sequence

Unk-Arg-Phe-NH2

Storage

Store at -20°C

Solubility

Soluble in DMSO, Water

InChI

InChI=1S/C26H38N6O3/c27-22(33)21(12-16-5-2-1-3-6-16)31-23(34)20(7-4-8-30-25(28)29)32-24(35)26-13-17-9-18(14-26)11-19(10-17)15-26/h1-3,5-6,17-21H,4,7-15H2,(H2,27,33)(H,31,34)(H,32,35)(H4,28,29,30)

InChI Key

UMKHUSRDQFQHAK-RNJMTYCLSA-N

Canonical SMILES

C1C2CC3CC1CC(C2)(C3)C(=O)NC(CCCN=C(N)N)C(=O)NC(CC4=CC=CC=C4)C(=O)N

1.Trifluoroacetic acid catalyzed highly regioselective bromocyclization of styrene-type carboxylic acid.

Chen T1, Yeung YY2. Org Biomol Chem. 2016 Apr 29. [Epub ahead of print]

A trifluoroacetic acid catalyzed highly 6-endo regioselective bromocyclization of styrene-type carboxylic acid has been developed. The resulting 3,4-dihydroisocoumarines are valuable building blocks in organic synthesis.