Found 111 with Last Name = 'abdel-rahman' and Initial = 'hm' TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Kyoto Pharmaceutical University
Curated by ChEMBL
Kyoto Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.00240nMAssay Description:Inhibition of HIV1 recombinant protease after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Kyoto Pharmaceutical University
Curated by ChEMBL
Kyoto Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.0310nMAssay Description:Inhibition of HIV1 recombinant protease after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
3D Structure (crystal)TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Kyoto Pharmaceutical University
Curated by ChEMBL
Kyoto Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Inhibition of HIV1 recombinant protease after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Kyoto Pharmaceutical University
Curated by ChEMBL
Kyoto Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 0.830nMAssay Description:Inhibition of HIV1 recombinant protease after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Inhibition of bovine brain mitochondria MAO-B using benzylamine substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 8.20nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of bovine brain mitochondria MAO-B using benzylamine substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of mouse full length GST-tagged BRAF V600E mutant using recombinant human His6-tagged MEK1 as substrate preincubated for 1 hr followed by ...More data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibition of bovine brain mitochondria MAO-B using benzylamine substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 64nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect ce...More data for this Ligand-Target Pair
Affinity DataIC50: 71nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 73nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 84nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 88nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 96nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 98nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:The compounds that exhibited potent anti-inflammatory profiles were futher tested for their ability to inhibit human COX-1 and COX-2 enzymes in-vitro...More data for this Ligand-Target Pair
Affinity DataIC50: <300nMAssay Description:The compounds that exhibited potent anti-inflammatory profiles were futher tested for their ability to inhibit human COX-1 and COX-2 enzymes in-vitro...More data for this Ligand-Target Pair
Affinity DataIC50: 780nMAssay Description:The compounds that exhibited potent anti-inflammatory profiles were futher tested for their ability to inhibit human COX-1 and COX-2 enzymes in-vitro...More data for this Ligand-Target Pair
Affinity DataIC50: 920nMAssay Description:The compounds that exhibited potent anti-inflammatory profiles were futher tested for their ability to inhibit human COX-1 and COX-2 enzymes in-vitro...More data for this Ligand-Target Pair
Affinity DataIC50: 930nMAssay Description:Inhibition of bovine brain mitochondria MAO-A using serotonin substrate after 60 mins by fluorimetric methodMore data for this Ligand-Target Pair
