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Found 47 with Last Name = 'abourbeh' and Initial = 'g'
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171516(CHEMBL363815 | N-[4-(4,5-Dichloro-2-fluoro-phenyla...)
Affinity DataIC50:  0.0400nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171514(2-Chloro-N-[4-(4,5-dichloro-2-fluoro-phenylamino)-...)
Affinity DataIC50:  0.0700nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171520((E)-4-Dimethylamino-but-2-enoic acid [4-(4,5-dichl...)
Affinity DataIC50:  0.110nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171525(2-Chloro-N-[4-(3-iodo-phenylamino)-quinazolin-6-yl...)
Affinity DataIC50:  0.120nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171523((4,5-Dichloro-2-fluoro-phenyl)-(6,7-dimethoxy-quin...)
Affinity DataIC50:  0.210nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM4583((2E)-N-{4-[(3-bromophenyl)amino]quinazolin-6-yl}-4...)
Affinity DataIC50:  0.410nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171524((E)-4-Dimethylamino-but-2-enoic acid [4-(3-iodo-ph...)
Affinity DataIC50:  0.940nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171520((E)-4-Dimethylamino-but-2-enoic acid [4-(4,5-dichl...)
Affinity DataIC50:  4nMAssay Description:Inhibition of HER1 kinase in intact DHER14 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171524((E)-4-Dimethylamino-but-2-enoic acid [4-(3-iodo-ph...)
Affinity DataIC50: <5nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171524((E)-4-Dimethylamino-but-2-enoic acid [4-(3-iodo-ph...)
Affinity DataIC50: <5nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171523((4,5-Dichloro-2-fluoro-phenyl)-(6,7-dimethoxy-quin...)
Affinity DataIC50:  5nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysate; Range = 3-5 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171518(CHEMBL193159 | N-[4-(3-Bromo-phenylamino)-quinazol...)
Affinity DataIC50: <5nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM4583((2E)-N-{4-[(3-bromophenyl)amino]quinazolin-6-yl}-4...)
Affinity DataIC50:  10nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysate; Range = 1-10 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171518(CHEMBL193159 | N-[4-(3-Bromo-phenylamino)-quinazol...)
Affinity DataIC50:  10nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM4583((2E)-N-{4-[(3-bromophenyl)amino]quinazolin-6-yl}-4...)
Affinity DataIC50:  10nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysate; Range = 1-10 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171525(2-Chloro-N-[4-(3-iodo-phenylamino)-quinazolin-6-yl...)
Affinity DataIC50:  10nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysate; Range = 4-10 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171520((E)-4-Dimethylamino-but-2-enoic acid [4-(4,5-dichl...)
Affinity DataIC50:  10nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysate; Range = 4-10 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171514(2-Chloro-N-[4-(4,5-dichloro-2-fluoro-phenylamino)-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of HER1 kinase in intact DHER14 cells; Range = 5-15 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171516(CHEMBL363815 | N-[4-(4,5-Dichloro-2-fluoro-phenyla...)
Affinity DataIC50:  20nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysate; Range = 6.7-20 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171516(CHEMBL363815 | N-[4-(4,5-Dichloro-2-fluoro-phenyla...)
Affinity DataIC50:  20nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysate; Range = 6.7-20 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171514(2-Chloro-N-[4-(4,5-dichloro-2-fluoro-phenylamino)-...)
Affinity DataIC50:  25nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysate; Range = 25-50 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171514(2-Chloro-N-[4-(4,5-dichloro-2-fluoro-phenylamino)-...)
Affinity DataIC50:  25nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysate; Range = 5-25 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171525(2-Chloro-N-[4-(3-iodo-phenylamino)-quinazolin-6-yl...)
Affinity DataIC50:  30nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171518(CHEMBL193159 | N-[4-(3-Bromo-phenylamino)-quinazol...)
Affinity DataIC50:  32nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171520((E)-4-Dimethylamino-but-2-enoic acid [4-(4,5-dichl...)
Affinity DataIC50:  50nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysate; Range = 10-50 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171514(2-Chloro-N-[4-(4,5-dichloro-2-fluoro-phenylamino)-...)
Affinity DataIC50:  50nMAssay Description:Inhibition of HER2 kinase in intact CSH12 cells; Range = 25-50 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171520((E)-4-Dimethylamino-but-2-enoic acid [4-(4,5-dichl...)
Affinity DataIC50:  50nMAssay Description:Inhibition of HER2 kinase in intact CSH12 cells; Range = 25-50 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171522(CHEMBL190567 | N-[4-(3-Iodo-phenylamino)-quinazoli...)
Affinity DataIC50:  150nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171521(CHEMBL192737 | N-[4-(3-Bromo-phenylamino)-quinazol...)
Affinity DataIC50:  174nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171515(CHEMBL190651 | N-[4-(4,5-Dichloro-2-fluoro-phenyla...)
Affinity DataIC50: >250nMAssay Description:Inhibition of HER1 kinase in intact DHER14 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171517(CHEMBL372246 | N-[4-(4,5-Dichloro-2-fluoro-phenyla...)
Affinity DataIC50:  250nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171519(CHEMBL365805 | N-[4-(3-Bromo-phenylamino)-7-(4-met...)
Affinity DataIC50:  250nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysate; Range = 50-250 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171515(CHEMBL190651 | N-[4-(4,5-Dichloro-2-fluoro-phenyla...)
Affinity DataIC50:  252nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171519(CHEMBL365805 | N-[4-(3-Bromo-phenylamino)-7-(4-met...)
Affinity DataIC50: >500nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171517(CHEMBL372246 | N-[4-(4,5-Dichloro-2-fluoro-phenyla...)
Affinity DataIC50: >500nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171515(CHEMBL190651 | N-[4-(4,5-Dichloro-2-fluoro-phenyla...)
Affinity DataIC50: >500nMAssay Description:Inhibition of HER2 kinase in intact CSH12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171514(2-Chloro-N-[4-(4,5-dichloro-2-fluoro-phenylamino)-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human PDGFR kinase in intact NIHPDGFR cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171515(CHEMBL190651 | N-[4-(4,5-Dichloro-2-fluoro-phenyla...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human PDGFR kinase in intact NIHPDGFR cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171520((E)-4-Dimethylamino-but-2-enoic acid [4-(4,5-dichl...)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human PDGFR kinase in intact NIHPDGFR cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171522(CHEMBL190567 | N-[4-(3-Iodo-phenylamino)-quinazoli...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysate; Range = 1000-5000 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171517(CHEMBL372246 | N-[4-(4,5-Dichloro-2-fluoro-phenyla...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171515(CHEMBL190651 | N-[4-(4,5-Dichloro-2-fluoro-phenyla...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysate; Range = 1000-10000 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171519(CHEMBL365805 | N-[4-(3-Bromo-phenylamino)-7-(4-met...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171521(CHEMBL192737 | N-[4-(3-Bromo-phenylamino)-quinazol...)
Affinity DataIC50: >1.30E+4nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171515(CHEMBL190651 | N-[4-(4,5-Dichloro-2-fluoro-phenyla...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysate; Range = 10000-50000 nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171522(CHEMBL190567 | N-[4-(3-Iodo-phenylamino)-quinazoli...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Hadassah Hebrew University

Curated by ChEMBL
LigandPNGBDBM50171521(CHEMBL192737 | N-[4-(3-Bromo-phenylamino)-quinazol...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of EGF Receptor autophosphorylation in A431 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed