Affinity DataKi: 0.700nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 4.10nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 5.20nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 72nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 91nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 115nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 132nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 399nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 436nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 463nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 601nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 935nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 1.52E+3nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 2.24E+3nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 5.82E+3nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 1.26E+4nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: 3.31E+4nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: 3.68E+4nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to Yersinia pestis ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
TargetThreonine--tRNA ligase 1, cytoplasmic(Homo sapiens (Human))
Trius Therapeutics
Curated by ChEMBL
Trius Therapeutics
Curated by ChEMBL
Affinity DataKi: >5.00E+4nMAssay Description:Binding affinity to human cytoplasmic ThrRS by coupled spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Inhibition of Aurora kinase A autophosphorylation in human HEK293 cells after 2 hrs by phosphor antibody readout assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Displacement of Alexa Fluor labelled kinase tracer178 from WEE1 (unknown origin) incubated for 60 mins by FRET assayMore data for this Ligand-Target Pair