Affinity DataKi: 140nMAssay Description:Inhibition of [3H] colchicine binding to bovine brain tubulin incubated for 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Inhibition of [3H] colchicine binding to bovine brain tubulin incubated for 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 260nMAssay Description:Inhibition of [3H] colchicine binding to bovine brain tubulin incubated for 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi
Curated by ChEMBL
University Of Karachi
Curated by ChEMBL
Affinity DataKi: 440nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi
Curated by ChEMBL
University Of Karachi
Curated by ChEMBL
Affinity DataKi: 850nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi
Curated by ChEMBL
University Of Karachi
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
Affinity DataKi: 2.20E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi
Curated by ChEMBL
University Of Karachi
Curated by ChEMBL
Affinity DataKi: 4.00E+3nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
Affinity DataKi: 4.20E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
Affinity DataKi: 4.50E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
Affinity DataKi: 4.60E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
Affinity DataKi: 5.00E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi
Curated by ChEMBL
University Of Karachi
Curated by ChEMBL
Affinity DataKi: 7.60E+3nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
Affinity DataKi: 8.00E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi
Curated by ChEMBL
University Of Karachi
Curated by ChEMBL
Affinity DataKi: 1.26E+4nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi
Curated by ChEMBL
University Of Karachi
Curated by ChEMBL
Affinity DataKi: 1.61E+4nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi
Curated by ChEMBL
University Of Karachi
Curated by ChEMBL
Affinity DataKi: 1.70E+4nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
Affinity DataKi: 1.80E+4nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi
Curated by ChEMBL
University Of Karachi
Curated by ChEMBL
Affinity DataKi: 2.06E+4nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi
Curated by ChEMBL
University Of Karachi
Curated by ChEMBL
Affinity DataKi: 2.55E+4nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
Affinity DataKi: 3.16E+4nMAssay Description:Inhibition of histamine N-methyltransferase in guinea pig brain using S-adenosyl-L-methionine-14C as substrate by scintillation spectrophotometerMore data for this Ligand-Target Pair
Affinity DataKi: 2.47E+5nMAssay Description:Inhibition of histamine N-methyltransferase in guinea pig brain using S-adenosyl-L-methionine-14C as substrate by scintillation spectrophotometerMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 6.60nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Egyptian National Research Centre
Curated by ChEMBL
Egyptian National Research Centre
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production using arachidonic acid as substrate preincubated with enzyme for 10 mins follo...More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production using arachidonic acid as substrate preincubated with enzyme for 10 mins follo...More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production using arachidonic acid as substrate preincubated with enzyme for 10 mins follo...More data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production using arachidonic acid as substrate preincubated with enzyme for 10 mins follo...More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production using arachidonic acid as substrate preincubated with enzyme for 10 mins follo...More data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Egyptian National Research Centre
Curated by ChEMBL
Egyptian National Research Centre
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of PDGFRbeta (unknown origin)More data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1/2/3/4(Homo sapiens (Human))
Egyptian National Research Centre
Curated by ChEMBL
Egyptian National Research Centre
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of FGFR (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
TargetFibroblast growth factor receptor 1/2/3/4(Homo sapiens (Human))
Egyptian National Research Centre
Curated by ChEMBL
Egyptian National Research Centre
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of FGFR (unknown origin)More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Egyptian National Research Centre
Curated by ChEMBL
Egyptian National Research Centre
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production using arachidonic acid as substrate preincubated with enzyme for 10 mins follo...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
National Research Centre
Curated by ChEMBL
National Research Centre
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair