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Found 42 with Last Name = 'akué-gédu' and Initial = 'r'
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50326438(9-trifluoromethyl-1,10-dihydropyrrolo[2,3-a]carbaz...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50326436(6-Bromo-1,10-dihydropyrrolo[2,3-a]carbazole-3-carb...)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50365178(CHEMBL1950228)
Affinity DataIC50:  8nMAssay Description:Inhibition of human recombinant His6-tagged PIM1 expressed in Sf21 cells using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50299249(1,10-Dihydropyrrolo[2,3-a]carbazole-3-carbaldehyde...)
Affinity DataIC50:  10nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50299249(1,10-Dihydropyrrolo[2,3-a]carbazole-3-carbaldehyde...)
Affinity DataIC50:  10nMAssay Description:Inhibition of Pim-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50326436(6-Bromo-1,10-dihydropyrrolo[2,3-a]carbazole-3-carb...)
Affinity DataIC50:  12.4nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50365178(CHEMBL1950228)
Affinity DataIC50:  13nMAssay Description:Inhibition of human recombinant His6-tagged PIM3 expressed in Sf21 cells using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50326438(9-trifluoromethyl-1,10-dihydropyrrolo[2,3-a]carbaz...)
Affinity DataIC50:  18nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50326441(9-Bromo-1,10-dihydropyrrolo[2,3-a]carbazole-3-carb...)
Affinity DataIC50:  24nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50326439(CHEMBL1243128 | Methyl 3-formyl-1,10-dihydropyrrol...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50326441(9-Bromo-1,10-dihydropyrrolo[2,3-a]carbazole-3-carb...)
Affinity DataIC50:  31nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50326439(CHEMBL1243128 | Methyl 3-formyl-1,10-dihydropyrrol...)
Affinity DataIC50:  40nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50299245(7-Bromo-1,10-dihydropyrrolo[2,3-a]carbazole-3-carb...)
Affinity DataIC50:  40nMAssay Description:Inhibition of Pim-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50385115(CHEMBL2036116)
Affinity DataIC50:  41nMAssay Description:Inhibition of Pim-3 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50385115(CHEMBL2036116)
Affinity DataIC50:  46nMAssay Description:Inhibition of Pim-1 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50326440(9-Ethyl-1,10-dihydropyrrolo[2,3-a]carbazole-3-carb...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50326440(9-Ethyl-1,10-dihydropyrrolo[2,3-a]carbazole-3-carb...)
Affinity DataIC50:  66nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50385117(CHEMBL2036118)
Affinity DataIC50:  75nMAssay Description:Inhibition of Pim-1 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50385117(CHEMBL2036118)
Affinity DataIC50:  80nMAssay Description:Inhibition of Pim-3 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50326437(8-Bromo-1,10-dihydropyrrolo[2,3-a]carbazole-3-carb...)
Affinity DataIC50:  90nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50365179(CHEMBL1950229)
Affinity DataIC50:  105nMAssay Description:Inhibition of human recombinant His6-tagged PIM1 expressed in Sf21 cells using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50365179(CHEMBL1950229)
Affinity DataIC50:  108nMAssay Description:Inhibition of human recombinant His6-tagged PIM3 expressed in Sf21 cells using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50326442(8-Methyl-1,10-dihydropyrrolo[2,3-a]carbazole-3-car...)
Affinity DataIC50:  117nMAssay Description:Inhibition of human GST fused Pim3 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50299249(1,10-Dihydropyrrolo[2,3-a]carbazole-3-carbaldehyde...)
Affinity DataIC50:  120nMAssay Description:Inhibition of Pim-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50299249(1,10-Dihydropyrrolo[2,3-a]carbazole-3-carbaldehyde...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human GST fused Pim1 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50326436(6-Bromo-1,10-dihydropyrrolo[2,3-a]carbazole-3-carb...)
Affinity DataIC50:  131nMAssay Description:Inhibition of human GST fused Pim2 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50299247(1-(1,10-Dihydropyrrolo[2,3-a]carbazol-3-yl)-2,2,2-...)
Affinity DataIC50:  170nMAssay Description:Inhibition of Pim-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50299250(7-(2,4-Difluorophenyl)-1,10-dihydropyrrolo[2,3-a]c...)
Affinity DataIC50:  200nMAssay Description:Inhibition of Pim-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50385116(CHEMBL2036117)
Affinity DataIC50:  200nMAssay Description:Inhibition of Pim-3 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50299248(1,10-Dihydropyrrolo[2,3-a]carbazole-3-carboxamide ...)
Affinity DataIC50:  210nMAssay Description:Inhibition of Pim-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50365180(CHEMBL1950230)
Affinity DataIC50:  235nMAssay Description:Inhibition of human recombinant His6-tagged PIM3 expressed in Sf21 cells using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50365180(CHEMBL1950230)
Affinity DataIC50:  315nMAssay Description:Inhibition of human recombinant His6-tagged PIM1 expressed in Sf21 cells using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50365181(CHEMBL1950358)
Affinity DataIC50:  327nMAssay Description:Inhibition of human recombinant His6-tagged PIM1 expressed in Sf21 cells using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50365178(CHEMBL1950228)
Affinity DataIC50:  350nMAssay Description:Inhibition of human recombinant PIM2 expressed in Escherichia coli using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50299246(7-Bromo-1,10-dihydropyrrolo[2,3-a]carbazole | CHEM...)
Affinity DataIC50:  440nMAssay Description:Inhibition of Pim-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50385116(CHEMBL2036117)
Affinity DataIC50:  470nMAssay Description:Inhibition of Pim-1 using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50365181(CHEMBL1950358)
Affinity DataIC50:  490nMAssay Description:Inhibition of human recombinant His6-tagged PIM3 expressed in Sf21 cells using RSRHSSYPAGT as substrate after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50299249(1,10-Dihydropyrrolo[2,3-a]carbazole-3-carbaldehyde...)
Affinity DataIC50:  510nMAssay Description:Inhibition of human GST fused Pim2 expressed in Escherichia coli after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50299249(1,10-Dihydropyrrolo[2,3-a]carbazole-3-carbaldehyde...)
Affinity DataIC50:  510nMAssay Description:Inhibition of Pim-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50299245(7-Bromo-1,10-dihydropyrrolo[2,3-a]carbazole-3-carb...)
Affinity DataIC50:  570nMAssay Description:Inhibition of Pim-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50299250(7-(2,4-Difluorophenyl)-1,10-dihydropyrrolo[2,3-a]c...)
Affinity DataIC50:  660nMAssay Description:Inhibition of Pim-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Clermont Université

Curated by ChEMBL
LigandPNGBDBM50299248(1,10-Dihydropyrrolo[2,3-a]carbazole-3-carboxamide ...)
Affinity DataIC50:  780nMAssay Description:Inhibition of Pim-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed