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Found 85 with Last Name = 'al-najjar' and Initial = 'bo'
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50336780(CHEMBL1672103 | sodium 1-amino-4-(3-amino-2-methyl...)
Affinity DataKi:  25nMAssay Description:Binding affinity to human P2Y12 expressed in astrocytoma cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50268918(1-Amino-2-methyl-4-[4-phenylamino-3-sulfophenylami...)
Affinity DataKi:  51nMAssay Description:Binding affinity to human P2Y12 expressed in astrocytoma cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50237558(CHEMBL1671994)
Affinity DataKi:  63nMAssay Description:Binding affinity to human P2Y12 expressed in astrocytoma cellsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50233805(CHEMBL4077922 | US11021454, Compound Salvianolic a...)
Affinity DataKi:  1.56E+4nMAssay Description:Displacement of [3H]2MeSADP from human P2Y12 expressed in U2OS cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50414250(CHEMBL457077)
Affinity DataKi:  2.03E+4nMAssay Description:Displacement of [3H]2MeSADP from human P2Y1 expressed in U2OS cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50587725(CHEMBL1615434)
Affinity DataKi:  3.64E+4nMAssay Description:Displacement of [3H]2MeSADP from human P2Y12 expressed in U2OS cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50594691(CHEMBL5176593)
Affinity DataIC50:  0.330nMAssay Description:Inhibition of 2-MeS-ADP induced P2Y12 (unknown origin) signalling expressed in CHO cells membrane incubated for 45 mins by 35S-GTPgammaS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50594686(CHEMBL5195237)
Affinity DataIC50:  1nMAssay Description:Displacement of tritium-labeled 2MeSADP from human P2Y12 expressed in CHO cells measured after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50594688(CHEMBL5192953)
Affinity DataIC50:  1nMAssay Description:Displacement of tritium-labeled 2MeSADP from human P2Y12 expressed in CHO cells measured after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50594687(CHEMBL5173489)
Affinity DataIC50:  1nMAssay Description:Displacement of tritium-labeled 2MeSADP from human P2Y12 expressed in CHO cells measured after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50594685(CHEMBL5184268)
Affinity DataIC50:  1nMAssay Description:Displacement of tritium-labeled 2MeSADP from human P2Y12 expressed in CHO cells measured after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50594684(CHEMBL5179719)
Affinity DataIC50:  1nMAssay Description:Displacement of tritium-labeled 2MeSADP from human P2Y12 expressed in CHO cells measured after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50594689(CHEMBL5203416)
Affinity DataIC50:  1nMAssay Description:Displacement of tritium-labeled 2MeSADP from human P2Y12 expressed in CHO cells measured after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50594682(CHEMBL5196387)
Affinity DataIC50:  2.80nMAssay Description:Displacement of tritium-labeled 2MeSADP from human P2Y12 expressed in CHO cells measured after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50594681(CHEMBL5188874)
Affinity DataIC50:  3nMAssay Description:Displacement of tritium-labeled 2MeSADP from human P2Y12 expressed in CHO cells measured after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM119428(US8669266, 679)
Affinity DataIC50:  3nMAssay Description:Displacement of [33P]2MeSADP from human P2Y12 expressed in CHO cell membranes preincubated for 15 mins followed by [33P]2MeSADP addition and measured...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50594678(CHEMBL5190693)
Affinity DataIC50:  10nMAssay Description:Displacement of [33P]2MeSADP from human P2Y12 expressed in CHO cell membranes preincubated for 15 mins followed by [33P]2MeSADP addition and measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50594677(CHEMBL5207212)
Affinity DataIC50:  10nMAssay Description:Displacement of [33P]2MeSADP from human P2Y12 expressed in CHO cell membranes preincubated for 15 mins followed by [33P]2MeSADP addition and measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50133663(5-{3-[3-(4-Benzoyl-2-propyl-phenoxy)-propoxy]-phen...)
Affinity DataIC50:  19nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50131514(5-(3-{3-[4-(4-Hydroxy-phenoxy)-2-propyl-phenoxy]-p...)
Affinity DataIC50:  30nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50133661(5-{3-[3-(4-Benzo[d]isoxazol-3-yl-2-propyl-phenoxy)...)
Affinity DataIC50:  30nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50594679(CHEMBL5170672)
Affinity DataIC50:  30nMAssay Description:Displacement of [33P]2MeSADP from human P2Y12 expressed in CHO cell membranes preincubated for 15 mins followed by [33P]2MeSADP addition and measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50594683(CHEMBL5204363)
Affinity DataIC50:  34nMAssay Description:Displacement of tritium-labeled 2MeSADP from human P2Y12 expressed in CHO cells measured after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50133658(5-{3-[3-(4-Cyclohexyloxy-2-propyl-phenoxy)-propoxy...)
Affinity DataIC50:  37nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50133654(5-{3-[3-(4-Cyclohexanecarbonyl-2-propyl-phenoxy)-p...)
Affinity DataIC50:  46nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50126019(CHEMBL1783033 | CHEMBL23874 | {3-Chloro-4-[3-(3-hy...)
Affinity DataIC50:  48nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50397204(ELINOGREL)
Affinity DataIC50:  50nMAssay Description:Displacement of [3H]2MeSADP from human P2Y12 preincubated for 5 mins followed by [3H]2MeSADP addition and measured after 15 mins by scintillation cou...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50131512(5-(3-{3-[4-(4-Chloro-3-methyl-phenoxy)-2-propyl-ph...)
Affinity DataIC50:  56nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50131503(5-{3-[3-(4-Phenoxy-2-propyl-phenoxy)-propoxy]-phen...)
Affinity DataIC50:  57nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50131503(5-{3-[3-(4-Phenoxy-2-propyl-phenoxy)-propoxy]-phen...)
Affinity DataIC50:  57nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50133666(5-{3-[3-(4-Cyclohexylmethyl-2-propyl-phenoxy)-prop...)
Affinity DataIC50:  59nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50594680(CHEMBL5207480)
Affinity DataIC50:  61nMAssay Description:Displacement of tritium-labeled 2MeSADP from human P2Y12 expressed in CHO cells measured after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50133667(5-{3-[3-(4-Cyclopentyloxy-2-propyl-phenoxy)-propox...)
Affinity DataIC50:  63nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50131511(5-(3-{3-[4-(3,4-Dichloro-phenoxy)-2-propyl-phenoxy...)
Affinity DataIC50:  64nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50302669((S)-5-(4-(butoxycarbonyl)piperazin-1-yl)-5-oxo-4-(...)
Affinity DataIC50:  71nMAssay Description:Displacement of tritium-labeled 2MeSADP from human P2Y12 expressed in CHO cells measured after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50131504(5-(3-{3-[4-(4-Chloro-phenoxy)-2-propyl-phenoxy]-pr...)
Affinity DataIC50:  73nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50131502(5-{3-[3-(4-Phenoxy-phenoxy)-propoxy]-phenyl}-thiaz...)
Affinity DataIC50:  76nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50131506(5-(3-{3-[4-(4-Fluoro-phenoxy)-2-propyl-phenoxy]-pr...)
Affinity DataIC50:  77nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50131505(5-(3-{3-[4-(4-Fluoro-3-methyl-phenoxy)-2-propyl-ph...)
Affinity DataIC50:  78nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50133669(5-{3-[3-(4-Cycloheptyloxy-2-propyl-phenoxy)-propox...)
Affinity DataIC50:  85nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50085040(CHEMBL278994 | L-796449 | {3-Chloro-4-[3-(3-phenyl...)
Affinity DataIC50:  94nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Al-Ahliyya Amman University

Curated by ChEMBL
LigandPNGBDBM50594693(CHEMBL5187308)
Affinity DataIC50:  100nMAssay Description:Inhibition of 2-MeS-ADP induced P2Y12 (unknown origin) signalling expressed in CHO cells membrane incubated for 45 mins by 35S-GTPgammaS assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50126016(2-(3-chloro-4-(3-(3-ethyl-7-propylbenzo[d]isoxazol...)
Affinity DataIC50:  110nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50126018(2-(3-chloro-4-(3-(7-propyl-3-(trifluoromethyl)benz...)
Affinity DataIC50:  140nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50133656(5-(3-{3-[4-(4-Chloro-benzoyl)-2-propyl-phenoxy]-pr...)
Affinity DataIC50:  144nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50346490((S)-5-(3-(3-(4-(cyclohexylidenemethyl)-2-propylphe...)
Affinity DataIC50:  150nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50131509(5-(3-{3-[4-(4-Isopropyl-phenoxy)-2-propyl-phenoxy]...)
Affinity DataIC50:  170nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50346507((S)-5-(3-(3-(4-((1r,4r)-4-hydroxycyclohexyl)-2-pro...)
Affinity DataIC50:  180nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50127931(5-{4-[3-(4-Phenoxy-2-propyl-phenoxy)-propoxy]-phen...)
Affinity DataIC50:  180nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universiti Sains Malaysia

Curated by ChEMBL
LigandPNGBDBM50131501(5-{3-[4-(4-Phenoxy-2-propyl-phenoxy)-butoxy]-pheny...)
Affinity DataIC50:  195nMAssay Description:Displacement of radio-labeled full agonist from PPARgamma receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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