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Found 68 with Last Name = 'allen' and Initial = 'ee'
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50041969(3-{2-Butyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  0.100nMAssay Description:Displacement of [125I]-Sar1-Ile8-AII (without BSA) from type 1 Angiotensin II receptor of rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281950(1-{2-Butyl-4-oxo-3-[2'-(2H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  0.5nMAssay Description:Displacement of [125I]-Sar1-Ile8-AII (without BSA) from type 1 Angiotensin II receptor of rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281953(1-{2-Butyl-4-oxo-3-[2'-(2H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  0.580nMAssay Description:Displacement of [125I]-Sar1-Ile8-AII (without BSA) from type 1 Angiotensin II receptor of rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281950(1-{2-Butyl-4-oxo-3-[2'-(2H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  0.75nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281964(CHEMBL25315 | {2-Butyl-4-oxo-3-[2'-(2H-tetrazol-5-...)
Affinity DataIC50:  0.830nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281962(2-Butyl-6-methanesulfinyl-3-[2'-(2H-tetrazol-5-yl)...)
Affinity DataIC50:  0.900nMAssay Description:Displacement of [125I]-Sar1-Ile8-AII (without BSA) from type 1 Angiotensin II receptor of rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281962(2-Butyl-6-methanesulfinyl-3-[2'-(2H-tetrazol-5-yl)...)
Affinity DataIC50:  1nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281966(CHEMBL25056 | Isopropyl-carbamic acid 2-butyl-4-ox...)
Affinity DataIC50:  1nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281938(2-Butyl-6-methyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [125I]-Sar1-Ile8-AII (without BSA) from type 1 Angiotensin II receptor of rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281949(6-Benzylamino-2-butyl-3-[2'-(2H-tetrazol-5-yl)-bip...)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [125I]-Sar1-Ile8-AII (without BSA) from type 1 Angiotensin II receptor of rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281929(6-Amino-2-butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-...)
Affinity DataIC50:  1.30nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281929(6-Amino-2-butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-...)
Affinity DataIC50:  1.30nMAssay Description:Binding affinity against Angiotensin II type 1 Receptor in rabbit aortic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50041970(CHEMBL280526 | {2-Butyl-4-oxo-3-[2'-(2H-tetrazol-5...)
Affinity DataIC50:  1.60nMAssay Description:Displacement of [125I]-Sar1-Ile8-AII (without BSA) from type 1 Angiotensin II receptor of rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50041963(CHEMBL24861 | {2-Butyl-4-oxo-3-[2'-(1H-tetrazol-5-...)
Affinity DataIC50:  1.60nMAssay Description:Displacement of [125I]-Sar1-Ile8-AII (without BSA) from type 1 Angiotensin II receptor of rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281967(2-Butyl-6-methylamino-3-[2'-(2H-tetrazol-5-yl)-bip...)
Affinity DataIC50:  2nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281927(CHEMBL281846 | Pentanoic acid {2-butyl-4-oxo-3-[2'...)
Affinity DataIC50:  2nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281927(CHEMBL281846 | Pentanoic acid {2-butyl-4-oxo-3-[2'...)
Affinity DataIC50:  2nMAssay Description:Binding affinity against Angiotensin II type 1 Receptor in rabbit aortic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281948(2-Butyl-6-methanesulfonyl-3-[2'-(2H-tetrazol-5-yl)...)
Affinity DataIC50:  3nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50041963(CHEMBL24861 | {2-Butyl-4-oxo-3-[2'-(1H-tetrazol-5-...)
Affinity DataIC50:  3.40nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281947(2-Butyl-6-ethyl-3-[2'-(2H-tetrazol-5-yl)-biphenyl-...)
Affinity DataIC50:  4nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281938(2-Butyl-6-methyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  4nMAssay Description:Binding affinity against Angiotensin II type 1 Receptor in rabbit aortic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281959(2-Butyl-6-isopropyl-3-[2'-(2H-tetrazol-5-yl)-biphe...)
Affinity DataIC50:  4nMAssay Description:Displacement of [125I]-Sar1-Ile8-AII (without BSA) from type 1 Angiotensin II receptor of rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281938(2-Butyl-6-methyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  4nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281946(CHEMBL282236 | {2-Butyl-4-oxo-3-[2'-(2H-tetrazol-5...)
Affinity DataIC50:  4.30nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281934(2-Butyl-6-methoxy-3-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataIC50:  5nMAssay Description:Binding affinity against Angiotensin II type 1 Receptor in rabbit aortic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281965(2-Butyl-6-pyridin-2-yl-3-[2'-(2H-tetrazol-5-yl)-bi...)
Affinity DataIC50:  5nMAssay Description:Displacement of [125I]-Sar1-Ile8-AII (without BSA) from type 1 Angiotensin II receptor of rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281959(2-Butyl-6-isopropyl-3-[2'-(2H-tetrazol-5-yl)-biphe...)
Affinity DataIC50:  5nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281955(2-Butyl-6-dimethylamino-3-[2'-(2H-tetrazol-5-yl)-b...)
Affinity DataIC50:  5nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281934(2-Butyl-6-methoxy-3-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataIC50:  5nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281945(2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50:  6nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281939(6-Methyl-2-pentyl-3-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataIC50:  6.40nMAssay Description:Binding affinity against Angiotensin II type 1 Receptor in rabbit aortic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50041970(CHEMBL280526 | {2-Butyl-4-oxo-3-[2'-(2H-tetrazol-5...)
Affinity DataIC50:  6.40nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281952(2-Butyl-6-methylsulfanyl-3-[2'-(2H-tetrazol-5-yl)-...)
Affinity DataIC50:  7nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281948(2-Butyl-6-methanesulfonyl-3-[2'-(2H-tetrazol-5-yl)...)
Affinity DataIC50:  7.60nMAssay Description:Displacement of [125I]-Sar1-Ile8-AII (without BSA) from type 1 Angiotensin II receptor of rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281949(6-Benzylamino-2-butyl-3-[2'-(2H-tetrazol-5-yl)-bip...)
Affinity DataIC50:  8nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281927(CHEMBL281846 | Pentanoic acid {2-butyl-4-oxo-3-[2'...)
Affinity DataIC50:  8.90nMAssay Description:Displacement of [125I]-Sar1-Ile8-AII (without BSA) from type 1 Angiotensin II receptor of rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281940(CHEMBL277182 | N-{2-Butyl-4-oxo-3-[2'-(1H-tetrazol...)
Affinity DataIC50:  9nMAssay Description:Binding affinity against Angiotensin II type 1 Receptor in rabbit aortic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281940(CHEMBL277182 | N-{2-Butyl-4-oxo-3-[2'-(1H-tetrazol...)
Affinity DataIC50:  9nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281945(2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50:  10nMAssay Description:Binding affinity against Angiotensin II type 1 Receptor in rabbit aortic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281943(6-Methyl-2-propyl-3-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataIC50:  10nMAssay Description:Binding affinity against Angiotensin II type 1 Receptor in rabbit aortic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281932(2-Butyl-5-fluoro-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  10nMAssay Description:Binding affinity against Angiotensin II type 1 Receptor in rabbit aortic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281942(2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmeth...)
Affinity DataIC50:  12nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from Angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281930(2-Butyl-6-iodo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4...)
Affinity DataIC50:  12nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from Angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281930(2-Butyl-6-iodo-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4...)
Affinity DataIC50:  12nMAssay Description:Displacement of [125I]-Sar1-Ile8-AII (without BSA) from type 1 Angiotensin II receptor of rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281937(2-Butyl-6,7-dimethoxy-3-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataIC50:  13nMAssay Description:Binding affinity against Angiotensin II type 1 Receptor in rabbit aortic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281937(2-Butyl-6,7-dimethoxy-3-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataIC50:  13nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281925(2-Butyl-7-chloro-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  15nMAssay Description:Binding affinity against Angiotensin II type 1 Receptor in rabbit aortic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281954(4'-{4-Oxo-3-[2'-(2H-tetrazol-5-yl)-biphenyl-4-ylme...)
Affinity DataIC50:  20nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281941(2-Butyl-6-fluoro-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  26nMAssay Description:Ability to displace [125I]-Sar1-Ile8-AII from angiotensin II receptor, type 1 in rabbit aorta in presence of 0.2% bovine serum albumin (BSA) was dete...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM50281941(2-Butyl-6-fluoro-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50:  26nMAssay Description:Binding affinity against Angiotensin II type 1 Receptor in rabbit aortic tissueMore data for this Ligand-Target Pair
In DepthDetails Article
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