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Found 318 with Last Name = 'altieri' and Initial = 'f'
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473413(CHEMBL126487)
Affinity DataKi:  2.30nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473417(CHEMBL129827)
Affinity DataKi:  4.5nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473417(CHEMBL129827)
Affinity DataKi:  4.5nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473414(CHEMBL129790)
Affinity DataKi:  6.80nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473414(CHEMBL129790)
Affinity DataKi:  6.80nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473431(CHEMBL128610)
Affinity DataKi:  8nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473437(CHEMBL126197)
Affinity DataKi:  22nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473450(CHEMBL125353)
Affinity DataKi:  22nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473437(CHEMBL126197)
Affinity DataKi:  22nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469866(CHEMBL46193)
Affinity DataKi:  23nMAssay Description:The compound is evaluated for binding affinity against central muscarinic receptor by using [3H]- QNB as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473447(CHEMBL131467)
Affinity DataKi:  40nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469864(CHEMBL3084476)
Affinity DataKi:  50nMAssay Description:Binding affinity for [3H]QNB in membrane preparations from rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Istituto Tumori&Quot;Giovanni Paolo Ii&Quot

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]rosiglitazone from N-terminal His-tagged human PPARgamma ligand binding domain expressed in Escherichia coli BL21 DE3 cells by sc...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50053616(4-(3-Chloro-phenyl)-1,1-dimethyl-piperazin-1-ium |...)
Affinity DataKi:  80nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50475680(Arecaidine Propargyl Ester)
Affinity DataKi:  87nMAssay Description:Binding affinity to cloned human muscarinic M2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Istituto Tumori&Quot;Giovanni Paolo Ii&Quot

Curated by ChEMBL
LigandPNGBDBM28762((2R)-2-(4-{2-[1,3-benzoxazol-2-yl(heptyl)amino]eth...)
Affinity DataKi:  88nMAssay Description:Displacement of [3H]rosiglitazone from N-terminal His-tagged human PPARgamma ligand binding domain expressed in Escherichia coli BL21 DE3 cells by sc...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473439(CHEMBL126517)
Affinity DataKi:  90nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473451(CHEMBL125357)
Affinity DataKi:  90nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469865(CHEMBL1160156)
Affinity DataKi:  95nMAssay Description:Binding affinity for [3H]QNB in membrane preparations from rat brain tissueMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469863(CHEMBL1160131)
Affinity DataKi:  110nMAssay Description:Binding affinity for [3H]QNB in membrane preparations from rat brain tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473430(CHEMBL126348)
Affinity DataKi:  170nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50006611(CHEMBL45951)
Affinity DataKi:  174nMAssay Description:The compound is evaluated for binding affinity against central muscarinic receptor by using [3H]- QNB as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50097722(CHEMBL129399)
Affinity DataKi:  180nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50061567(1,1-Dimethyl-4-phenyl-piperazin-1-ium | CHEMBL1347...)
Affinity DataKi:  250nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473469(CHEMBL126452)
Affinity DataKi:  300nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473434(CHEMBL337220)
Affinity DataKi:  386nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473470(CHEMBL128847)
Affinity DataKi:  420nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473416(CHEMBL126030)
Affinity DataKi:  500nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473412(CHEMBL125636)
Affinity DataKi:  600nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473412(CHEMBL125636)
Affinity DataKi:  603nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473459(CHEMBL129266)
Affinity DataKi:  644nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473458(CHEMBL129232)
Affinity DataKi:  672nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473453(CHEMBL129772)
Affinity DataKi:  750nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473453(CHEMBL129772)
Affinity DataKi:  759nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473418(CHEMBL341158)
Affinity DataKi:  794nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473418(CHEMBL341158)
Affinity DataKi:  800nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473423(CHEMBL125904)
Affinity DataKi:  850nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50475680(Arecaidine Propargyl Ester)
Affinity DataKi:  851nMAssay Description:Binding affinity to cloned human muscarinic M3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473468(CHEMBL128682)
Affinity DataKi:  851nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473468(CHEMBL128682)
Affinity DataKi:  853nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473445(CHEMBL129291)
Affinity DataKi:  900nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50475680(Arecaidine Propargyl Ester)
Affinity DataKi:  933nMAssay Description:Binding affinity to cloned human muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Istituto Tumori&Quot;Giovanni Paolo Ii&Quot

Curated by ChEMBL
LigandPNGBDBM28763((2S)-2-(4-{2-[1,3-benzoxazol-2-yl(heptyl)amino]eth...)
Affinity DataKi:  971nMAssay Description:Displacement of [3H]rosiglitazone from N-terminal His-tagged human PPARgamma ligand binding domain expressed in Escherichia coli BL21 DE3 cells by sc...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50475680(Arecaidine Propargyl Ester)
Affinity DataKi:  977nMAssay Description:Binding affinity to cloned human muscarinic M4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473425(CHEMBL127023)
Affinity DataKi:  1.02E+3nMAssay Description:compound was evaluated for pKiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473425(CHEMBL127023)
Affinity DataKi:  1.03E+3nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473463(1'',2'',3'',6''-Tetrahydro-[3,4'']Bipyridinyl HCl ...)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50473433(CHEMBL542222)
Affinity DataKi:  1.20E+3nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50053627(1,1-Dimethyl-4-(3-trifluoromethyl-phenyl)-piperazi...)
Affinity DataKi:  1.20E+3nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rattus norvegicus (Rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50026638(1'-Methyl-1',2',3',6'-tetrahydro-[3,4']bipyridinyl...)
Affinity DataKi:  1.20E+3nMAssay Description:Binding affinity against nicotinic receptors from rat brain using [3H]cystine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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