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Found 29 with Last Name = 'amblard' and Initial = 'mc'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286545(3-Benzenesulfonyl-5-chloro-2-(1H-imidazol-2-yl)-1H...)
Affinity DataIC50:  3.5nMAssay Description:Inhibitory activity against HIV-1 RT with poly.rC-oligo.dG template primerMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50230553(3-Benzenesulfonyl-5-chloro-2-(5-methyl-1H-imidazol...)
Affinity DataIC50:  4.70nMAssay Description:Inhibitory activity against HIV-1 RT with poly.rC-oligo.dG template primerMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286549(3-Benzenesulfonyl-5-chloro-2-(4,5-dimethyl-1H-imid...)
Affinity DataIC50:  5.10nMAssay Description:Inhibitory activity against HIV-1 RT with poly.rC-oligo.dG template primerMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286550(3-Benzenesulfonyl-5-chloro-2-(4,5-dihydro-1H-imida...)
Affinity DataIC50:  6.5nMAssay Description:Inhibitory activity against HIV-1 RT with poly.rC-oligo.dG template primerMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286551(2-(3-Benzenesulfonyl-5-chloro-1H-indol-2-yl)-4,5,6...)
Affinity DataIC50:  8.10nMAssay Description:Inhibitory activity against HIV-1 RT with poly.rC-oligo.dG template primerMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50230553(3-Benzenesulfonyl-5-chloro-2-(5-methyl-1H-imidazol...)
Affinity DataIC50:  9nMAssay Description:Inhibitory activity against K103N mutant of HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286543(3-Benzenesulfonyl-5-chloro-2-(4-methyl-5-propyl-1H...)
Affinity DataIC50:  9.40nMAssay Description:Inhibitory activity against HIV-1 RT with poly.rC-oligo.dG template primerMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286548(3-Benzenesulfonyl-5-chloro-2-(4,5-diethyl-1H-imida...)
Affinity DataIC50:  10nMAssay Description:Inhibitory activity against HIV-1 RT with poly.rC-oligo.dG template primerMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286542(3-Benzenesulfonyl-5-chloro-2-(4,5-dihydro-thiazol-...)
Affinity DataIC50:  17nMAssay Description:Inhibitory activity against HIV-1 RT with poly.rC-oligo.dG template primerMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286546(4-(3-Benzenesulfonyl-5-chloro-1H-indol-2-yl)-4H-1l...)
Affinity DataIC50:  20nMAssay Description:Inhibitory activity against HIV-1 RT with poly.rC-oligo.dG template primerMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286549(3-Benzenesulfonyl-5-chloro-2-(4,5-dimethyl-1H-imid...)
Affinity DataIC50:  22nMAssay Description:Inhibitory activity against HIV-2 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286545(3-Benzenesulfonyl-5-chloro-2-(1H-imidazol-2-yl)-1H...)
Affinity DataIC50:  23nMAssay Description:Inhibitory activity against HIV-2 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286552((3aS,7aS)-2-(3-Benzenesulfonyl-5-chloro-1H-indol-2...)
Affinity DataIC50:  29nMAssay Description:Inhibitory activity against HIV-1 RT with poly.rC-oligo.dG template primerMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286544(3-Benzenesulfonyl-5-chloro-2-(5,5-dimethyl-4,5-dih...)
Affinity DataIC50:  50nMAssay Description:Inhibitory activity against HIV-1 RT with poly.rC-oligo.dG template primerMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286543(3-Benzenesulfonyl-5-chloro-2-(4-methyl-5-propyl-1H...)
Affinity DataIC50:  210nMAssay Description:Inhibitory activity against HIV-2 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286546(4-(3-Benzenesulfonyl-5-chloro-1H-indol-2-yl)-4H-1l...)
Affinity DataIC50:  222nMAssay Description:Inhibitory activity against K103N mutant of HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286550(3-Benzenesulfonyl-5-chloro-2-(4,5-dihydro-1H-imida...)
Affinity DataIC50:  358nMAssay Description:Inhibitory activity against HIV-2 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286545(3-Benzenesulfonyl-5-chloro-2-(1H-imidazol-2-yl)-1H...)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibitory activity against K103N/Y181C double mutant of HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286542(3-Benzenesulfonyl-5-chloro-2-(4,5-dihydro-thiazol-...)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibitory activity against K103N mutant of HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286547(3-Benzenesulfonyl-5-chloro-2-(1,4,5,6-tetrahydro-p...)
Affinity DataIC50:  2.29E+3nMAssay Description:Inhibitory activity against HIV-1 RT with poly.rC-oligo.dG template primerMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286553(3-Benzenesulfonyl-5-chloro-2-imidazol-1-yl-1H-indo...)
Affinity DataIC50:  2.39E+3nMAssay Description:Inhibitory activity against HIV-1 RT with poly.rC-oligo.dG template primerMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286549(3-Benzenesulfonyl-5-chloro-2-(4,5-dimethyl-1H-imid...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory activity against K103N/Y181C double mutant of HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286545(3-Benzenesulfonyl-5-chloro-2-(1H-imidazol-2-yl)-1H...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibitory activity against HIV-2 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286542(3-Benzenesulfonyl-5-chloro-2-(4,5-dihydro-thiazol-...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibitory activity against K103N mutant of HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286549(3-Benzenesulfonyl-5-chloro-2-(4,5-dimethyl-1H-imid...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibitory activity against K103N mutant of HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286550(3-Benzenesulfonyl-5-chloro-2-(4,5-dihydro-1H-imida...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibitory activity against HIV-2 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286543(3-Benzenesulfonyl-5-chloro-2-(4-methyl-5-propyl-1H...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibitory activity against HIV-2 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50230553(3-Benzenesulfonyl-5-chloro-2-(5-methyl-1H-imidazol...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibitory activity against K103N mutant of HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50286546(4-(3-Benzenesulfonyl-5-chloro-1H-indol-2-yl)-4H-1l...)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibitory activity against K103N mutant of HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails Article