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Found 12 with Last Name = 'amici' and Initial = 'l'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yale University

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataIC50:  0.0750nMAssay Description:In vivo binding affinity of the compound against dopamine (D2) receptor in rat caudate-putamen tissue using [3H]-nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Yale University

Curated by ChEMBL
LigandPNGBDBM79172(2-[4-[(3Z)-3-[2-(trifluoromethyl)-9-thioxanthenyli...)
Affinity DataIC50:  0.300nMAssay Description:In vivo binding affinity of the compound against dopamine (D1) receptor in rat caudate-putamen tissue using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yale University

Curated by ChEMBL
LigandPNGBDBM50012961((-)-(S)-N-((1-ethylpyrrolidin-2-yl)methyl)-2-hydro...)
Affinity DataIC50:  1.20nMAssay Description:In vivo inhibitory activity of the compound against dopamine (D1) receptor in rat caudate-putamen tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Yale University

Curated by ChEMBL
LigandPNGBDBM50012961((-)-(S)-N-((1-ethylpyrrolidin-2-yl)methyl)-2-hydro...)
Affinity DataIC50:  1.20nMAssay Description:In vivo binding affinity of the compound against dopamine (D1) receptor in rat caudate-putamen tissue using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yale University

Curated by ChEMBL
LigandPNGBDBM50012961((-)-(S)-N-((1-ethylpyrrolidin-2-yl)methyl)-2-hydro...)
Affinity DataIC50:  1.70nMAssay Description:In vivo inhibitory activity of the compound against dopamine (D2) receptor in rat caudate-putamen tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yale University

Curated by ChEMBL
LigandPNGBDBM50005118((S)-3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)...)
Affinity DataIC50:  7.20nMAssay Description:In vivo inhibitory activity of the compound against dopamine (D2) receptor in rat caudate-putamen tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yale University

Curated by ChEMBL
LigandPNGBDBM50007534(3-Bromo-N-((S)-1-ethyl-pyrrolidin-2-ylmethyl)-2-hy...)
Affinity DataIC50:  21nMAssay Description:In vivo inhibitory activity of the compound against dopamine (D2) receptor in rat caudate-putamen tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yale University

Curated by ChEMBL
LigandPNGBDBM50026561(3-Bromo-N-((S)-1-ethyl-pyrrolidin-2-ylmethyl)-6-hy...)
Affinity DataIC50:  56nMAssay Description:In vivo inhibitory activity of the compound against dopamine (D2) receptor in rat caudate-putamen tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Yale University

Curated by ChEMBL
LigandPNGBDBM50135412(CHEMBL423331 | N-((S)-1-Ethyl-pyrrolidin-2-ylmethy...)
Affinity DataIC50:  196nMAssay Description:In vivo inhibitory activity of the compound against dopamine (D2) receptor in rat caudate-putamen tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Yale University

Curated by ChEMBL
LigandPNGBDBM50012961((-)-(S)-N-((1-ethylpyrrolidin-2-yl)methyl)-2-hydro...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vivo binding affinity of the compound against dopamine (D2) receptor in rat caudate-putamen tissue using [3H]-nemonapride as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Yale University

Curated by ChEMBL
LigandPNGBDBM50135412(CHEMBL423331 | N-((S)-1-Ethyl-pyrrolidin-2-ylmethy...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vivo inhibitory activity of the compound against dopamine (D1) receptor in rat caudate-putamen tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Yale University

Curated by ChEMBL
LigandPNGBDBM50005118((S)-3,5-Dichloro-N-(1-ethyl-pyrrolidin-2-ylmethyl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vivo inhibitory activity of the compound against dopamine (D1) receptor in rat caudate-putamen tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed