Compile Data Set for Download or QSAR
maximum 50k data
Found 613 with Last Name = 'anand' and Initial = 's'
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50276625(1-Adamantan-1-yl-3-[3-(3-morpholin-4-yl-propoxy)-p...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of soluble epoxide hydrolase (unknown origin) by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50276625(1-Adamantan-1-yl-3-[3-(3-morpholin-4-yl-propoxy)-p...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human soluble epoxide hydrolase by fluorescent endpoint assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50296210(1-Adamantan-1-yl-3-[4-fluoro-3-(3-morpholin-4-yl-p...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human soluble epoxide hydrolase by fluorescent endpoint assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM25743(1-cycloheptyl-3-(1-acetylpiperidin-4-yl)urea | US8...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human soluble epoxide hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50296223(1-(4-(3-morpholinopropoxy)phenyl)-3-(4-(trifluorom...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human soluble epoxide hydrolase by fluorescent endpoint assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50296224(1-(4-(3-morpholinopropoxy)phenyl)-3-(4-(trifluorom...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human soluble epoxide hydrolase by fluorescent endpoint assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50296214(1-(4-fluoro-3-(3-morpholinopropoxy)phenyl)-3-(4-(t...)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of human soluble epoxide hydrolase by fluorescent endpoint assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM234969(US9556148, 40 | n-(cyanomethyl)-4-(5-methyl-2-((4-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human JAK1 kinase domainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50276673(1-(3-(3-morpholinopropoxy)phenyl)-3-(4-(trifluorom...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human soluble epoxide hydrolase by fluorescent endpoint assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317315(1-(3-(3-morpholinopropylsulfonyl)phenyl)-3-(4-(tri...)
Affinity DataIC50:  1nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317313(1-(3-(morpholinosulfonyl)phenyl)-3-(4-(trifluorome...)
Affinity DataIC50:  1nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317312(CHEMBL1099390 | N-(2-morpholinoethyl)-3-(3-(4-(tri...)
Affinity DataIC50:  1nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317310(1-(4-(3-morpholinopropylsulfonyl)phenyl)-3-(4-(tri...)
Affinity DataIC50:  1nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317308(1-(4-(morpholinosulfonyl)phenyl)-3-(4-(trifluorome...)
Affinity DataIC50:  1nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317290(CHEMBL1086820 | N-(2-morpholinoethyl)-4-(3-(4-(tri...)
Affinity DataIC50:  1nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM50600312(CHEMBL5189266)
Affinity DataIC50:  1nMAssay Description:Inhibition of human JAK1 kinase domainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50276673(1-(3-(3-morpholinopropoxy)phenyl)-3-(4-(trifluorom...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of soluble epoxide hydrolase (unknown origin) by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50296226(2-Adamantan-1-yl-N-[4-(3-morpholin-4-yl-propoxy)-p...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human soluble epoxide hydrolase by fluorescent endpoint assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50296213(1-(4-fluoro-3-(3-morpholinopropoxy)phenyl)-3-(4-(t...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human soluble epoxide hydrolase by fluorescent endpoint assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50223389(1-Adamantan-1-yl-3-[4-(3-morpholin-4-yl-propoxy)-p...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of human soluble epoxide hydrolase by fluorescent endpoint assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50296225(1-(4-chlorophenyl)-3-(4-(3-morpholinopropoxy)pheny...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human soluble epoxide hydrolase by fluorescent endpoint assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50335965(1-(1-(isopropylsulfonyl)piperidin-4-yl)-3-(4-(trif...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of human soluble epoxide hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50335964(1-(1-nicotinoylpiperidin-4-yl)-3-(4-(trifluorometh...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of human soluble epoxide hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50523667(CHEMBL4560054)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of human PI3Kdelta using PIP2 as substrate after 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50335966(1-Adamantan-1-yl-3-(1-methanesulfonyl-piperidin-4-...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of human soluble epoxide hydrolaseMore data for this Ligand-Target Pair
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317305(1-(3-fluoro-4-(morpholine-4-carbonyl)phenyl)-3-(4-...)
Affinity DataIC50:  2nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50296197(1-(4-chlorophenyl)-3-(3-(3-morpholinopropoxy)pheny...)
Affinity DataIC50:  2nMAssay Description:Inhibition of human soluble epoxide hydrolase by fluorescent endpoint assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317303(2-fluoro-N-(2-morpholinoethyl)-4-(3-(4-(trifluorom...)
Affinity DataIC50:  2nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317291(CHEMBL1086821 | N-(2-morpholinoethyl)-4-(3-(4-(tri...)
Affinity DataIC50:  2nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317282(1-(4-(4-isopropylpiperazine-1-carbonyl)phenyl)-3-(...)
Affinity DataIC50:  2nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50403068(CHEMBL2216870 | IDELALISIB | US9745321, CAL-101)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of human PI3Kdelta using PIP2 as substrate after 1 hrMore data for this Ligand-Target Pair
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50296219(1-Adamantan-1-yl-3-[3-(3-morpholin-4-yl-propoxy)-c...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of human soluble epoxide hydrolase by fluorescent endpoint assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50276676(2-Adamantan-1-yl-N-[3-(3-morpholin-4-yl-propoxy)-p...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of human soluble epoxide hydrolase by fluorescent endpoint assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50276676(2-Adamantan-1-yl-N-[3-(3-morpholin-4-yl-propoxy)-p...)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of soluble epoxide hydrolase (unknown origin) by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50335967(1-(1-(isopropylsulfonyl)piperidin-4-yl)-3-(4-(trif...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of human soluble epoxide hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM234969(US9556148, 40 | n-(cyanomethyl)-4-(5-methyl-2-((4-...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human JAK2 kinase domainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Cadila Healthcare

Curated by ChEMBL
LigandPNGBDBM50600312(CHEMBL5189266)
Affinity DataIC50:  3nMAssay Description:Inhibition of human JAK2 kinase domainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317286(4-{[(adamantan-1-yl)carbamoyl]amino}-N-[2-(morphol...)
Affinity DataIC50:  3nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317299(CHEMBL1087492 | N-(2-morpholino-2-oxoethyl)-4-(3-(...)
Affinity DataIC50:  3nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317307(CHEMBL1088351 | N-(2-morpholinoethyl)-4-(3-(4-(tri...)
Affinity DataIC50:  3nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317311(1-(3-(4-isopropylpiperazin-1-ylsulfonyl)phenyl)-3-...)
Affinity DataIC50:  3nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Mus musculus (Mouse))
Ar£Te Therapeutics

Curated by ChEMBL
LigandPNGBDBM50191854(CHEMBL436774 | N-(1-acetyl-piperidin-4-yl)-N'-(ada...)
Affinity DataIC50:  3nMAssay Description:Inhibition of mouse soluble epoxide hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50335968(1-(1-(methylsulfonyl)piperidin-4-yl)-3-(4-(trifluo...)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of human soluble epoxide hydrolaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50335966(1-Adamantan-1-yl-3-(1-methanesulfonyl-piperidin-4-...)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of soluble epoxide hydrolase in HUVEC assessed inhibition of as conversion of 14, 15-EET to 14, 15-DHETMore data for this Ligand-Target Pair
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50276626(1-cyclohexyl-3-(3-(3-morpholinopropoxy)phenyl)urea...)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of soluble epoxide hydrolase (unknown origin) by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50276626(1-cyclohexyl-3-(3-(3-morpholinopropoxy)phenyl)urea...)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of human soluble epoxide hydrolase by fluorescent endpoint assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317298(1-(4-(morpholine-4-carbonyl)phenyl)-3-(4-(trifluor...)
Affinity DataIC50:  4nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317301(1-(3-fluoro-4-(4-methylpiperazine-1-carbonyl)pheny...)
Affinity DataIC50:  4nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional epoxide hydrolase 2(Homo sapiens (Human))
ArêTe Therapeutics

Curated by ChEMBL
LigandPNGBDBM50317283(1-(4-(4-isopropylpiperazine-1-carbonyl)phenyl)-3-(...)
Affinity DataIC50:  4nMAssay Description:Inhibition of soluble epoxide hydrolase by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50523668(CHEMBL4550603)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of human PI3Kdelta using PIP2 as substrate after 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 613 total ) | Next | Last >>
Jump to: