Affinity DataKi: 0.110nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.320nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.330nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.660nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 0.710nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibitory constant against human coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibitory constant against human coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibitory constant against human coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Inhibitory constant against human coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 4.30nMAssay Description:Displacement of [3H]haTRAP from PAR1 in human platelet membraneMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]haTRAP from PAR-1 receptor in human platelet membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibitory constant against human coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibitory constant against human coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 8.40nMAssay Description:Inhibitory constant against human coagulation factor Xa (fXa)More data for this Ligand-Target Pair
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 8.90nMAssay Description:Displacement of [3H]haTRAP from PAR-1 receptor in human platelet membranes after 1 hr by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibitory constant against human coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute
Curated by ChEMBL
Schering-Plough Research Institute
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]haTRAP from PAR1 in human platelet membraneMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition constant against human factor XaMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibitory constant against human coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibitory constant against human coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Compound was tested for inhibition activity against Coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibitory constant against human coagulation factor Xa (fXa)More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Inhibitory potency was measured against human coagulation factor XMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Inhibitory constant against human coagulation factor Xa (fXa)More data for this Ligand-Target Pair