Affinity DataIC50: 0.310nMAssay Description:Binding affinity was measured against Opioid receptor delta 1 using [3H]-p-Cl-DPDPE as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 1.06nMAssay Description:Binding affinity was measured against Opioid receptor delta 1 using [3H]-p-Cl-DPDPE as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Binding affinity was measured against cloned human Opioid receptor delta 1 (wild-type,Wt)More data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Binding affinity was measured against mutated human Opioid receptor delta 1 (W248L)More data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Binding affinity was measured against Opioid receptor delta 1 using [3H]-p-Cl-DPDPE as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMAssay Description:Binding affinity was measured against Opioid receptor delta 1 using [3H]-p-Cl-DPDPE as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:Binding affinity was measured against cloned human Opioid receptor delta 1 (wild-type,Wt)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity was measured against Opioid receptor delta 1 using [3H]-p-Cl-DPDPE as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:In vitro inhibition of [3H]-deltorphin binding to Opioid receptor delta 1 using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 5.5nMAssay Description:Binding affinity was measured against cloned human Opioid receptor delta 1 (wild-type,Wt)More data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:Binding affinity was measured against Opioid receptor delta 1 using [3H]-p-Cl-DPDPE as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:In vitro inhibition of [3H]-deltorphin binding to Opioid receptor delta 1 using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:Binding affinity was measured against Opioid receptor delta 1 using [3H]-p-Cl-DPDPE as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 9.70nMAssay Description:Binding affinity was measured against Opioid receptor mu 1 using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of [3H]-deltorphin binding to Opioid receptor delta 1 using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Binding affinity was measured against mutated human Opioid receptor delta 1 (W248L)More data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Binding affinity was measured against Opioid receptor delta 1 using [3H]-p-Cl-DPDPE as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:In vitro inhibition of [3H]-deltorphin binding to Opioid receptor delta 1 using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Binding affinity was measured against Opioid receptor delta 1 using [3H]-p-Cl-DPDPE as radioligand.More data for this Ligand-Target Pair
TargetPantetheinase(Homo sapiens (Human))
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of human serum vanin-1 using pantetheine-7-amino-4-trifluoromethykournarin as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:In vitro inhibition of [3H]-deltorphin binding to Opioid receptor delta 1 using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:In vitro inhibition of [3H]-deltorphin binding to Opioid receptor delta 1 using rat brain membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 49nMAssay Description:Binding affinity was measured against mutated human Opioid receptor delta 1 (W248L)More data for this Ligand-Target Pair
TargetPantetheinase(Homo sapiens (Human))
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human serum vanin-1 using pantetheine-7-amino-4-trifluoromethykournarin as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
TargetPantetheinase(Homo sapiens (Human))
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of human serum vanin-1 using pantetheine-7-amino-4-trifluoromethykournarin as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Binding affinity was measured against Opioid receptor delta 1 using [3H]-p-Cl-DPDPE as radioligand.More data for this Ligand-Target Pair
TargetPantetheinase(Homo sapiens (Human))
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of human serum vanin-1 using pantetheine-7-amino-4-trifluoromethykournarin as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Agonist activity of the compound was determined using electrically induced smooth muscle contraction of mouse vas deferens.More data for this Ligand-Target Pair
Affinity DataIC50: 390nMAssay Description:Agonist activity of the compound was determined using electrically induced smooth muscle contraction of mouse vas deferens.More data for this Ligand-Target Pair
TargetPantetheinase(Homo sapiens (Human))
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibition of human serum vanin-1 using pantetheine-7-amino-4-trifluoromethykournarin as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
Affinity DataIC50: 420nMAssay Description:Binding affinity was measured against Opioid receptor delta 1 using [3H]-p-Cl-DPDPE as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Binding affinity was measured against Opioid receptor mu 1 using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
TargetPantetheinase(Homo sapiens (Human))
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of human serum vanin-1 using pantetheine-7-amino-4-trifluoromethykournarin as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
Affinity DataIC50: 609nMAssay Description:Binding affinity was measured against Opioid receptor mu 1 using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 609nMAssay Description:Binding affinity was measured against Opioid receptor mu 1 using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 610nMAssay Description:Binding affinity was measured against Opioid receptor delta 1 using [3H]-p-Cl-DPDPE as radioligand.More data for this Ligand-Target Pair
TargetPantetheinase(Homo sapiens (Human))
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 770nMAssay Description:Inhibition of human serum vanin-1 using pantetheine-7-amino-4-trifluoromethykournarin as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
TargetPantetheinase(Homo sapiens (Human))
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 770nMAssay Description:Inhibition of human serum vanin-1 using pantetheine-7-amino-4-trifluoromethykournarin as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
Affinity DataIC50: 780nMAssay Description:Binding affinity was measured against Opioid receptor mu 1 using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
TargetPantetheinase(Homo sapiens (Human))
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 780nMAssay Description:Inhibition of human serum vanin-1 using pantetheine-7-amino-4-trifluoromethykournarin as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
TargetPantetheinase(Homo sapiens (Human))
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of human serum vanin-1 using pantetheine-7-amino-4-trifluoromethykournarin as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Binding affinity was measured against Opioid receptor delta 1 using [3H]-p-Cl-DPDPE as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Binding affinity was measured against Opioid receptor mu 1 using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 2.26E+3nMAssay Description:Agonist activity of the compound was determined using electrically induced smooth muscle contraction of mouse vas deferens.More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity was measured against Opioid receptor mu 1 using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
TargetPantetheinase(Homo sapiens (Human))
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Osaka Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.84E+3nMAssay Description:Inhibition of human serum vanin-1 using pantetheine-7-amino-4-trifluoromethykournarin as substrate preincubated for 10 mins followed by substrate add...More data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:In vitro inhibition of [3H]-DAMGO (Tyr-D-Ala-Gly-(Me)-Phe-Gly-ol) binding to Opioid receptor mu 1 using rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+3nMAssay Description:Binding affinity was measured against Opioid receptor mu 1 using [3H]-DAMGO as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+3nMAssay Description:In vitro inhibition of [3H]-DAMGO (Tyr-D-Ala-Gly-(Me)-Phe-Gly-ol) binding to Opioid receptor mu 1 using rat brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+3nMAssay Description:In vitro inhibition of [3H]-DAMGO (Tyr-D-Ala-Gly-(Me)-Phe-Gly-ol) binding to Opioid receptor mu 1 using rat brain membranesMore data for this Ligand-Target Pair