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Found 1573 with Last Name = 'palmer' and Initial = 'ws'
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408198(CHEMBL91278)
Affinity DataKi:  0.0794nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408201(CHEMBL88512)
Affinity DataKi:  0.126nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50060964((R)-5-(2-((2-(2-ethoxyphenoxy)ethyl)amino)propyl)-...)
Affinity DataKi:  0.126nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.126nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408246(CHEMBL92261)
Affinity DataKi:  0.398nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408248(CHEMBL330060)
Affinity DataKi:  0.398nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50033112(6-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyla...)
Affinity DataKi:  0.501nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50160165(CHEMBL88272 | RS-17053 | [2-(2-Cyclopropylmethoxy-...)
Affinity DataKi:  0.794nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408244(CHEMBL93736)
Affinity DataKi:  0.794nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408242(CHEMBL91876)
Affinity DataKi:  0.794nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408232(CHEMBL91093)
Affinity DataKi:  0.794nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM31046(3-[4,5-dihydro-1H-imidazol-2-ylmethyl-(4-methylphe...)
Affinity DataKi:  0.794nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408229(CHEMBL329160)
Affinity DataKi:  0.794nMAssay Description:The compound was screened in vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408205(CHEMBL88435)
Affinity DataKi:  0.794nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408239(CHEMBL90874)
Affinity DataKi:  1.60nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408202(CHEMBL92901)
Affinity DataKi:  1.60nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408208(CHEMBL88820)
Affinity DataKi:  1.60nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408238(CHEMBL89916)
Affinity DataKi:  1.60nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408192(CHEMBL90869)
Affinity DataKi:  1.60nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408194(CHEMBL90287)
Affinity DataKi:  2nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50033111(1-(4-Amino-6,7-dimethoxy-2-quinazolinyl)-4-((tetra...)
Affinity DataKi:  2.5nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408225(CHEMBL312935)
Affinity DataKi:  3.20nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408193(CHEMBL92109)
Affinity DataKi:  7.90nMAssay Description:In vitro for the displacement of [3H]prazosin binding to bovine Alpha-1A adrenergic receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408216(CHEMBL90746)
Affinity DataKi:  79nMAssay Description:The compound's binding affinity against Alpha-2B adrenergic receptor from rat kidney homogenate in the presence of phentolamineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408216(CHEMBL90746)
Affinity DataKi:  126nMAssay Description:The compound's binding affinity against Dopamine receptor D2Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408197(CHEMBL91605)
Affinity DataKi:  6.40E+3nMAssay Description:The compound's binding affinity against Dopamine receptor D2Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408197(CHEMBL91605)
Affinity DataKi:  6.50E+3nMAssay Description:The compound's binding affinity against 5-hydroxytryptamine 1A receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408236(CHEMBL420620)
Affinity DataKi:  6.50E+3nMAssay Description:The compound's binding affinity against Alpha-2B adrenergic receptor from rat kidney homogenate in the presence of phentolamineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408241(CHEMBL89030)
Affinity DataKi:  6.50E+3nMAssay Description:The compound's binding affinity against Alpha-2B adrenergic receptor from rat kidney homogenate in the presence of phentolamineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50394918(CHEMBL2165504)
Affinity DataKi:  6.60E+3nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomes preincubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408236(CHEMBL420620)
Affinity DataKi:  6.70E+3nMAssay Description:The compound's binding affinity against Dopamine receptor D2Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408236(CHEMBL420620)
Affinity DataKi:  6.70E+3nMAssay Description:The compound's binding affinity against 5-hydroxytryptamine 1A receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408241(CHEMBL89030)
Affinity DataKi:  7.30E+3nMAssay Description:The compound's binding affinity against Dopamine receptor D2Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408229(CHEMBL329160)
Affinity DataKi:  7.40E+3nMAssay Description:The compound's binding affinity against Dopamine receptor D2Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408199(CHEMBL88160)
Affinity DataKi:  7.50E+3nMAssay Description:The compound's binding affinity against 5-hydroxytryptamine 1A receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408229(CHEMBL329160)
Affinity DataKi:  7.60E+3nMAssay Description:The compound's binding affinity against 5-hydroxytryptamine 1A receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408241(CHEMBL89030)
Affinity DataKi:  8.00E+3nMAssay Description:The compound's binding affinity against 5-hydroxytryptamine 1A receptorChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408199(CHEMBL88160)
Affinity DataKi:  8.10E+3nMAssay Description:The compound's binding affinity against Dopamine receptor D2Checked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(NEONATAL RAT)
Roche Bioscience

Curated by ChEMBL
LigandPNGBDBM50408199(CHEMBL88160)
Affinity DataKi:  8.60E+3nMAssay Description:The compound's binding affinity against Alpha-2B adrenergic receptor from rat kidney homogenate in the presence of phentolamineChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Genentech

Curated by ChEMBL
LigandPNGBDBM50394917(CHEMBL2165505)
Affinity DataKi:  7.80E+4nMAssay Description:Time dependent inhibition of CYP3A4 in human liver microsomes preincubated for 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50394916(CHEMBL2165506)
Affinity DataIC50:  0.480nMAssay Description:Binding affinity to PI3Kdelta after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50394910(CHEMBL2165512)
Affinity DataIC50:  0.670nMAssay Description:Binding affinity to PI3Kdelta after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50394913(CHEMBL2165509)
Affinity DataIC50:  1.10nMAssay Description:Binding affinity to PI3Kdelta after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50394920(CHEMBL2165672)
Affinity DataIC50:  1.70nMAssay Description:Binding affinity to PI3Kdelta after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50394921(CHEMBL2165671)
Affinity DataIC50:  1.80nMAssay Description:Binding affinity to PI3Kdelta after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50394908(CHEMBL2165666)
Affinity DataIC50:  1.80nMAssay Description:Binding affinity to PI3Kdelta after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Roche Palo Alto

US Patent
LigandPNGBDBM102578(US8536172, I-27)
Affinity DataIC50:  2nMpH: 7.5Assay Description:JNK activity was measured by phosphorylation of GST-ATF2 (19-96) with [gamma-33P] ATP.More data for this Ligand-Target Pair
In DepthDetails US Patent
LigandPNGBDBM50394893(CHEMBL2165502)
Affinity DataIC50:  2.30nMAssay Description:Binding affinity to PI3Kdelta after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50394909(CHEMBL2165513)
Affinity DataIC50:  2.30nMAssay Description:Binding affinity to PI3Kdelta after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50394903(CHEMBL2165492)
Affinity DataIC50:  2.40nMAssay Description:Binding affinity to PI3Kdelta after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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