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Found 19 with Last Name = 'redburn' and Initial = 'j'
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]naloxone from mu opioid receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50381677(CHEMBL1256748 | U-69593)
Affinity DataIC50:  8nMAssay Description:Displacement of [3H]naloxone from kappa opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAspartate-semialdehyde dehydrogenase(Helicobacter pylori)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50269414(CHEMBL457665 | CYSTEINE-S-SULFONIC ACID | S-sulpho...)
Affinity DataIC50:  180nMAssay Description:Inhibition of Helicobacter pylori His-tagged ASD assessed as inhibition of phosphorylation of aspartate semialdehydeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50316549(CHEMBL1097805 | longanine)
Affinity DataIC50:  700nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50316551(CHEMBL1096481 | N-methylstephuline)
Affinity DataIC50:  2.10E+3nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50316546(CHEMBL1097077 | N-methylstephisoferulin)
Affinity DataIC50:  2.50E+3nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50269198(9alpha,11alpha-epoxycholest-7-ene-3beta,5alpha,6al...)
Affinity DataIC50:  4.50E+3nMAssay Description:Displacement of [125I]IL8 from human recombinant IL8 type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50316547(6-cinnamoylhernandine | CHEMBL1097804)
Affinity DataIC50:  5.10E+3nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50269197(CHEMBL451438 | cholest-8-ene-3beta,5alpha,6alpha,7...)
Affinity DataIC50:  5.50E+3nMAssay Description:Displacement of [125I]IL8 from human recombinant IL8 type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50316552(CHEMBL1096482 | prostephabyssine)
Affinity DataIC50:  5.50E+3nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50377943(LATIFOLIAN B)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of JNK3-induced transfer of [gamma33P]ATP to biotinylated ATF2 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50316545(6-cinnamoyl-N-methylstephasunoline | CHEMBL1098354)
Affinity DataIC50:  1.13E+4nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50377942(LATIFOLIAN A)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of JNK3-induced transfer of [gamma33P]ATP to biotinylated ATF2 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50316550(CHEMBL1097185 | aknadilactam)
Affinity DataIC50:  1.70E+4nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 1(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50269196(CHEMBL501985 | cholest-8-ene-3beta,5alpha,6alpha,7...)
Affinity DataIC50:  2.00E+4nMAssay Description:Displacement of [125I]IL8 from human recombinant IL8 type A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50260779(CHEMBL524026 | sinococuline)
Affinity DataIC50:  3.70E+4nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Griffith University

Curated by ChEMBL
LigandPNGBDBM50316548(CHEMBL1098359 | aknadinine)
Affinity DataIC50:  4.60E+4nMAssay Description:Displacement of [3H]deltorphin-2 from human delta opioid receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAspartate-semialdehyde dehydrogenase(Helicobacter pylori)
Griffith University

Curated by ChEMBL
LigandPNGBDBM50377941(PETROSAMINE B)
Affinity DataIC50:  3.06E+5nMAssay Description:Inhibition of Helicobacter pylori His-tagged ASD assessed as inhibition of phosphorylation of aspartate semialdehydeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed