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Found 258 with Last Name = 'rognan' and Initial = 'd'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50354644(CHEMBL1834218)
Affinity DataKi:  0.0250nMAssay Description:Displacement of [3H]DAMGO from rat brain Mu-type opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50354647(CHEMBL1834244)
Affinity DataKi:  0.0250nMAssay Description:Displacement of [3H]DAMGO from rat brain Mu-type opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50266025((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Affinity DataKi:  0.0310nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in Sprague-Dawley rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50354650(CHEMBL1834247)
Affinity DataKi:  0.0470nMAssay Description:Displacement of [3H]DAMGO from rat brain Mu-type opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50266025((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50354649(CHEMBL1834246)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]DAMGO from rat brain Mu-type opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50354651(CHEMBL1834248)
Affinity DataKi:  0.330nMAssay Description:Displacement of [3H]DAMGO from rat brain Mu-type opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50354645(CHEMBL1834219)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]DAMGO from rat brain Mu-type opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50189920((S)-2-amino-N-((S)-2-(2-(benzylamino)-2-oxoethyl)-...)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50354644(CHEMBL1834218)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]Ile-deltorphin-2 from rat brain delta-type opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFe(3+)-pyochelin receptor(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50444965(CHEMBL3099904)
Affinity DataKi:  2.20nMAssay Description:Displacement of Pch-55Fe(III) from Pseudomonas aeruginosa PAD07 FptA after 1 hr in presence of CCCPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50354650(CHEMBL1834247)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]Ile-deltorphin-2 from rat brain delta-type opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50266060((S)-2-amino-N-((R)-2-(2-(benzylamino)-2-oxoethyl)-...)
Affinity DataKi:  3.35nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50354648(CHEMBL1834245)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]DAMGO from rat brain Mu-type opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFe(3+)-pyochelin receptor(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50444963(CHEMBL3099907)
Affinity DataKi:  6.5nMAssay Description:Displacement of Pch-55Fe(III) from Pseudomonas aeruginosa PAD07 FptA after 1 hr in presence of CCCPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50266063(2-((S)-4-((S)-2-(dimethylamino)-3-(4-hydroxy-2,6-d...)
Affinity DataKi:  6.64nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in Sprague-Dawley rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFe(3+)-pyochelin receptor(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50444964(CHEMBL3099905)
Affinity DataKi:  9.80nMAssay Description:Displacement of Pch-55Fe(III) from Pseudomonas aeruginosa PAD07 FptA after 1 hr in presence of CCCPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50266026((S)-6-amino-2-((S)-4-((S)-2-amino-3-(4-hydroxy-2,6...)
Affinity DataKi:  10.1nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFe(3+)-pyochelin receptor(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
University Of Strasburg

Curated by ChEMBL
LigandPNGBDBM50444962(CHEMBL3099909)
Affinity DataKi:  11nMAssay Description:Displacement of Pch-55Fe(III) from Pseudomonas aeruginosa PAD07 FptA after 1 hr in presence of CCCPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50189920((S)-2-amino-N-((S)-2-(2-(benzylamino)-2-oxoethyl)-...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in Sprague-Dawley rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50266056((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-N-((S...)
Affinity DataKi:  12.4nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50354646(CHEMBL1834220)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]DAMGO from rat brain Mu-type opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50266057((S)-2-(dimethylamino)-3-(4-hydroxy-2,6-dimethylphe...)
Affinity DataKi:  20.5nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in Sprague-Dawley rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50354647(CHEMBL1834244)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]Ile-deltorphin-2 from rat brain delta-type opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369245(CHEMBL4170392)
Affinity DataKi:  25nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369246(CHEMBL4160309)
Affinity DataKi:  44nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369285(CHEMBL4160346)
Affinity DataKi:  48nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50266058((S)-2-amino-N-((S)-2-(2-(benzylamino)-2-oxoethyl)-...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369286(CHEMBL4167574)
Affinity DataKi:  53nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50042947(1-(4-Chloro-phenyl)-3-(4-hydroxy-3-methoxy-phenyl)...)
Affinity DataKi:  53nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50354649(CHEMBL1834246)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]Ile-deltorphin-2 from rat brain delta-type opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50266057((S)-2-(dimethylamino)-3-(4-hydroxy-2,6-dimethylphe...)
Affinity DataKi:  64.9nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369256(CHEMBL4175451)
Affinity DataKi:  71nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369250(CHEMBL4168923)
Affinity DataKi:  107nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369280(CHEMBL4166275)
Affinity DataKi:  107nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369248(CHEMBL4163005)
Affinity DataKi:  107nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369244(CHEMBL4169628)
Affinity DataKi:  107nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369321(CHEMBL4168220)
Affinity DataKi:  107nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50266061((S)-N-((R)-2-(2-(benzylamino)-2-oxoethyl)-3-oxo-1,...)
Affinity DataKi:  133nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50266060((S)-2-amino-N-((R)-2-(2-(benzylamino)-2-oxoethyl)-...)
Affinity DataKi:  161nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in Sprague-Dawley rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369330(CHEMBL4160583)
Affinity DataKi:  203nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50266059(CHEMBL501023 | benzyl 2-((S)-4-((S)-2-amino-3-(4-h...)
Affinity DataKi:  244nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369279(CHEMBL4166454)
Affinity DataKi:  267nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369249(CHEMBL4173832)
Affinity DataKi:  285nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50266026((S)-6-amino-2-((S)-4-((S)-2-amino-3-(4-hydroxy-2,6...)
Affinity DataKi:  290nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in Sprague-Dawley rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50354651(CHEMBL1834248)
Affinity DataKi:  337nMAssay Description:Displacement of [3H]Ile-deltorphin-2 from rat brain delta-type opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50042973(1-(4-Chloro-phenyl)-3-(3,4-dihydroxy-phenyl)-prope...)
Affinity DataKi:  350nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369292(CHEMBL4175213)
Affinity DataKi:  357nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369278(CHEMBL4162605)
Affinity DataKi:  357nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStromal cell-derived factor 1(Homo sapiens (Human))
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50369322(CHEMBL4170951)
Affinity DataKi:  357nMAssay Description:Binding affinity to Texas Red-labelled CXCL12 (unknown origin) assessed as inhibition of CXCL12-Texas Red binding to EGFP-labeled human CXCR4 express...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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