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Found 2162 with Last Name = 'roy' and Initial = 'r'
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50001885((risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  0.501nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50477152(CHEMBL393466)
Affinity DataKi:  0.643nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1 receptor in rat brainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50003020(MK-3102 | OMARIGLIPTIN | US10155775, Omarigliptin ...)
Affinity DataKi:  0.800nMAssay Description:Competitive reversible inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50304627((2S,3S,4R,5R,6S)-6-methylpiperidine-2,3,4,5-tetrao...)
Affinity DataKi:  1nMAssay Description:Inhibition of bovine kidney alpha-L-fucosidase by para-nitrophenolate release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50065258((2S,3R,4S,5R)-2-Methyl-piperidine-3,4,5-triol | (2...)
Affinity DataKi:  3nMAssay Description:Inhibition of bovine kidney alpha-L-fucosidase by para-nitrophenolate release assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50001885((risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50477152(CHEMBL393466)
Affinity DataKi:  9.40nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat brainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50304628((2S,3R,4S)-2-methyl-3,4-dihydro-2H-pyrrole-3,4-dio...)
Affinity DataKi:  10nMAssay Description:Inhibition of bovine kidney alpha-L-fucosidase by para-nitrophenolate release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50133931(1-(4-fluoro-phenyl)-4-(3,4,6,7,12,12a-hexahydro-1H...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50133931(1-(4-fluoro-phenyl)-4-(3,4,6,7,12,12a-hexahydro-1H...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  35nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50066974(7-Benzyl-2,3-dihydroxy-6-methyl-4-propyl-naphthale...)
Affinity DataKi:  50nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  58nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1 receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50477151(CHEMBL393622)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat brainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50477151(CHEMBL393622)
Affinity DataKi:  94nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat brainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50066979(2,3-Dihydroxy-6,7-dimethyl-4-propyl-naphthalene-1-...)
Affinity DataKi:  100nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50066979(2,3-Dihydroxy-6,7-dimethyl-4-propyl-naphthalene-1-...)
Affinity DataKi:  100nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50010449(3,4,3',4'-Tetrahydroxy-5,5'-diisopropyl-7,7'-dimet...)
Affinity DataKi:  150nMAssay Description:The compound was tested for inhibitory activity against aldose reductase from human placentaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50066975(7-Benzyl-2,3-dihydroxy-4-isopropyl-6-methyl-naphth...)
Affinity DataKi:  200nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50066973(2,3-Dihydroxy-4-isopropyl-6-methyl-7-(4-trifluorom...)
Affinity DataKi:  200nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50066974(7-Benzyl-2,3-dihydroxy-6-methyl-4-propyl-naphthale...)
Affinity DataKi:  300nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50010436(6,7,6',7'-Tetrahydroxy-5,5'-diisopropyl-1,1'-dimet...)
Affinity DataKi:  310nMAssay Description:The compound was tested for inhibitory activity against aldose reductase from human placentaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(RAT)
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50133931(1-(4-fluoro-phenyl)-4-(3,4,6,7,12,12a-hexahydro-1H...)
Affinity DataKi:  425nMAssay Description:Displacement of [3H]SCH-23390 from dopamine D1 receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50066976(7-Benzyl-2,3-dihydroxy-4,6-dimethyl-naphthalene-1-...)
Affinity DataKi:  500nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM23223(7-[8-formyl-1,6,7-trihydroxy-3-methyl-5-(propan-2-...)
Affinity DataKi:  500nMAssay Description:The compound was tested for inhibitory activity against Aldose reductase from human placentaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50066975(7-Benzyl-2,3-dihydroxy-4-isopropyl-6-methyl-naphth...)
Affinity DataKi:  700nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue alpha-L-fucosidase(Bos taurus)
Universit£

Curated by ChEMBL
LigandPNGBDBM50304626((2R,3S,4S,5S)-2-methylpiperidine-3,4,5-triol | CHE...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of bovine kidney alpha-L-fucosidase by para-nitrophenolate release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50066974(7-Benzyl-2,3-dihydroxy-6-methyl-4-propyl-naphthale...)
Affinity DataKi:  1.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-H)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50066981(2,3-Dihydroxy-4-isopropyl-6,7-dimethyl-naphthalene...)
Affinity DataKi:  1.00E+3nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50066977(2,3-Dihydroxy-6-methyl-4-propyl-naphthalene-1-carb...)
Affinity DataKi:  1.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50010451(But-2-enoic acid 1'-but-2-enoyloxy-8,8'-dicyano-6,...)
Affinity DataKi:  1.30E+3nMAssay Description:The compound was tested for inhibitory activity against Aldose reductase from human placentaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50010446(1,7,1',7'-Tetrahydroxy-5,5'-diisopropyl-6,6'-dimet...)
Affinity DataKi:  1.50E+3nMAssay Description:The compound was tested for inhibitory activity against Aldose reductase from human placentaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50066981(2,3-Dihydroxy-4-isopropyl-6,7-dimethyl-naphthalene...)
Affinity DataKi:  2.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50031638(2,3-Dihydroxy-4-isopropyl-6-methyl-naphthalene-1-c...)
Affinity DataKi:  2.00E+3nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Central Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50477152(CHEMBL393466)
Affinity DataKi:  2.25E+3nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat brainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50010437(2,2-Dimethyl-propionic acid 8,8'-dicyano-1'-(2,2-d...)
Affinity DataKi:  2.50E+3nMAssay Description:The compound was tested for inhibitory activity against Aldose reductase from human placentaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50010450(6,7,6',7'-Tetrahydroxy-5,5'-diisopropyl-1,1'-dimet...)
Affinity DataKi:  2.80E+3nMAssay Description:The compound was tested for inhibitory activity against Aldose reductase from human placentaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50031638(2,3-Dihydroxy-4-isopropyl-6-methyl-naphthalene-1-c...)
Affinity DataKi:  3.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50010440(CHEMBL326383 | Hexanoic acid 8,8'-dicyano-1'-hexan...)
Affinity DataKi:  3.10E+3nMAssay Description:The compound was tested for inhibitory activity against aldose reductase from human placentaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50066980(2,3-Dihydroxy-4,6,7-trimethyl-naphthalene-1-carbox...)
Affinity DataKi:  4.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-M)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50010447(8,8'-Bis-hydroxymethyl-5,5'-diisopropyl-1,1'-dimet...)
Affinity DataKi:  4.30E+3nMAssay Description:The compound was tested for inhibitory activity against Aldose reductase from human placentaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50010444(CHEMBL52639 | Pentanoic acid 8,8'-dicyano-6,7,6',7...)
Affinity DataKi:  4.70E+3nMAssay Description:The compound was tested for inhibitory activity against aldose reductase from human placentaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50010435(Butyric acid 1'-butyryloxy-8,8'-dicyano-6,7,6',7'-...)
Affinity DataKi:  5.30E+3nMAssay Description:The compound was tested for inhibitory activity against aldose reductase from human placentaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50066977(2,3-Dihydroxy-6-methyl-4-propyl-naphthalene-1-carb...)
Affinity DataKi:  6.00E+3nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50010439(CHEMBL297483 | Propionic acid 8,8'-dicyano-6,7,6',...)
Affinity DataKi:  6.80E+3nMAssay Description:The compound was tested for inhibitory activity against aldose reductase from human placentaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50066975(7-Benzyl-2,3-dihydroxy-4-isopropyl-6-methyl-naphth...)
Affinity DataKi:  7.00E+3nMAssay Description:inhibitory activity against Human Lactate Dehydrogenase (LDH-H)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50010438(Acetic acid 1'-acetoxy-8,8'-dicyano-6,7,6',7'-tetr...)
Affinity DataKi:  7.30E+3nMAssay Description:The compound was tested for inhibitory activity against aldose reductase from human placentaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldo-keto reductase family 1 member B1(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50229024(CHEMBL3349372)
Affinity DataKi:  7.80E+3nMAssay Description:The compound was tested for inhibitory activity against Aldose reductase from human placentaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
University Of New Mexico School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50066976(7-Benzyl-2,3-dihydroxy-4,6-dimethyl-naphthalene-1-...)
Affinity DataKi:  8.00E+3nMAssay Description:inhibitory activity against P. falciparum lactate dehydrogenase (pLDH)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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