Affinity DataKi: 18nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 61nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 290nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 1.50E+3nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 6.80E+3nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+4nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human Peroxisome proliferator activated recep...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined by displacement of 20 nM [3H]- thiazolidinedione from 4 nM biotinylated human peroxisome proliferator-activated recep...More data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Inhibition of ET-1 stimulated arachidonic acid release in rabbit renal vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of ET-1 stimulated arachidonic acid release in rabbit renal vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of ET-1 stimulated arachidonic acid release in CHO cells expressing rat ET- B receptorsMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of ET-1 stimulated arachidonic acid release in CHO cells expressing rat ET- B receptorsMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of ET-1 stimulated arachidonic acid release in rabbit renal vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of ET-1 stimulated arachidonic acid release in rabbit renal vascular smooth muscle cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
Affinity DataIC50: 37nMAssay Description:Binding affinity measured in CHO cells stably transfected with the human endothelin B receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Binding affinity against endothelin A receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Binding affinity against endothelin B receptor from rabbit renal vascular smooth musclesMore data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Binding affinity against endothelin B receptor rat cerebellar membranes.More data for this Ligand-Target Pair