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Found 46 with Last Name = 'shapiro' and Initial = 'hs'
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227363(CHEMBL299837)
Affinity DataKi:  0.100nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227366(CHEMBL48927)
Affinity DataKi:  0.200nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227361(CHEMBL51585)
Affinity DataKi:  0.25nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227364(CHEMBL299093)
Affinity DataKi:  0.25nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227640(CHEMBL297952)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227355(CHEMBL296821)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227356(CHEMBL49944)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227358(CHEMBL412056)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227365(CHEMBL300096)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227642(CHEMBL50562)
Affinity DataKi:  0.300nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50009073(4-(5-cyclopentyloxycarbonylamino-1-methyl-1H-indol...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015528(CHEMBL50370 | N-[3-(4-Benzenesulfonylaminocarbonyl...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015523(CHEMBL52492 | N-{4-[5-(3-Cyclopentyl-ureido)-1-pro...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000819(2-Cyclopentyl-N-{3-[2-methoxy-4-(toluene-2-sulfony...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227390(CHEMBL301616)
Affinity DataKi:  0.5nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227389(CHEMBL51580)
Affinity DataKi:  0.700nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015551(CHEMBL301498 | N-{4-[5-(3-Cyclopentyl-ureido)-1-me...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227367(CHEMBL48435)
Affinity DataKi:  0.800nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015517(2-Cyclopentyl-N-{3-[2-methoxy-4-(toluene-2-sulfony...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015540(CHEMBL431348 | N-{4-[5-(3-Cyclopentyl-ureido)-1-me...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227638(CHEMBL49566)
Affinity DataKi:  1.40nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50009070((2S,3R)-3-(2-Carboxy-ethylsulfanyl)-2-hydroxy-3-[2...)
Affinity DataKi:  5nMAssay Description:Inhibition constant for displasement of [3H]-LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227354(CHEMBL51289)
Affinity DataKi:  5.60nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227353(CHEMBL51239)
Affinity DataKi:  6.80nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227359(CHEMBL51061)
Affinity DataKi:  10nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015542(4-[5-Cyclopentyloxycarbonylamino-1-(2-methoxy-ethy...)
Affinity DataKi:  41nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015516(4-[6-(2-Cyclopentyl-acetylamino)-indazol-1-ylmethy...)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227357(CHEMBL49981)
Affinity DataKi:  53nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227360(CHEMBL50364)
Affinity DataKi:  57nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015539(4-(5-Cyclopentyloxycarbonylamino-1-propyl-1H-indol...)
Affinity DataKi:  58nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227391(CHEMBL430967)
Affinity DataKi:  67nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227362(CHEMBL300943)
Affinity DataKi:  70nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227641(CHEMBL297014)
Affinity DataKi:  71nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015521(4-[5-(2-Cyclopentyl-acetylamino)-1-methyl-1H-indol...)
Affinity DataKi:  80nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015544(4-(6-Cyclopentyloxycarbonylamino-indazol-1-ylmethy...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227639(CHEMBL52260)
Affinity DataKi:  84nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1/2(Homo sapiens (Human))
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50227352(CHEMBL300906)
Affinity DataKi:  132nMAssay Description:Inhibition constant for displacement of [3H]LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015529(4-(5-Cyclopentyloxycarbonylamino-1-methyl-1H-indol...)
Affinity DataKi:  157nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015525(4-(5-Cyclopentyloxycarbonylamino-1-methyl-1H-indaz...)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015549(4-(6-Cyclopentyloxycarbonylamino-indol-1-ylmethyl)...)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015520(4-[6-(2-Cyclopentyl-acetylamino)-indol-1-ylmethyl]...)
Affinity DataKi:  200nMAssay Description:Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015522(4-(5-Cyclopentyloxycarbonylamino-1H-indol-3-ylmeth...)
Affinity DataKi:  236nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015519(4-[5-(3-Cyclopentyl-ureido)-1-methyl-1H-indol-3-yl...)
Affinity DataKi:  1.12E+3nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015537(4-[5-(2-Ethyl-pentanoylamino)-1-methyl-1H-indol-3-...)
Affinity DataKi:  1.83E+3nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50015510(4-(5-Hexanoylamino-1-methyl-1H-indol-3-ylmethyl)-3...)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Ici Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50006816((LY-171883)1-{2-Hydroxy-3-propyl-4-[4-(1H-tetrazol...)
Affinity DataKi:  2.82E+3nMAssay Description:Displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed