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Found 227 with Last Name = 'shoji' and Initial = 'm'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50019290(CHEMBL3289390)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]NMS from human M2R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50377964(Cantil | Glycophenylate | MEPENZOLATE BROMIDE | Me...)
Affinity DataKi:  0.680nMAssay Description:Displacement of [3H]NMS from human M2R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50019290(CHEMBL3289390)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]NMS from human M3R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50019289(CHEMBL3289391)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]NMS from human M2R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50377964(Cantil | Glycophenylate | MEPENZOLATE BROMIDE | Me...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]NMS from human M3R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127501(3-(4-Carbamimidoyl-2-{2-[4-(pyrrolidine-1-carbonyl...)
Affinity DataKi:  3nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127492(4-[5-Carbamimidoyl-2-(2-carboxy-2-oxo-ethyl)-pheno...)
Affinity DataKi:  11nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127502(4-[5-Carbamimidoyl-2-(2-carboxy-2-oxo-ethyl)-pheno...)
Affinity DataKi:  18nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127495(3-[4-Carbamimidoyl-2-(2-{4-[1-(1-imino-ethyl)-pipe...)
Affinity DataKi:  20nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127504(CHEMBL55770 | N-[2-(3-Carbamimidoyl-phenoxy)-ethyl...)
Affinity DataKi:  20nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127494(3-(4-Carbamimidoyl-2-{2-[(3,4,5,6-tetrahydro-2H-[1...)
Affinity DataKi:  21nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127498(3-{4-Carbamimidoyl-2-[2-(4-carbamimidoyl-benzoylam...)
Affinity DataKi:  26nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50019289(CHEMBL3289391)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]NMS from human M3R expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127503(3-(4-Carbamimidoyl-benzoylamino)-4-(3-carbamimidoy...)
Affinity DataKi:  28nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127493(3-(4-Carbamimidoyl-2-{2-[(3,4,5,6-tetrahydro-2H-[1...)
Affinity DataKi:  43nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127506(3-(4-Carbamimidoyl-benzoylamino)-4-(3-carbamimidoy...)
Affinity DataKi:  170nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127496(CHEMBL51796 | N-[2-(3-Carbamimidoyl-phenoxy)-ethyl...)
Affinity DataKi:  170nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127497(4-Carbamimidoyl-N-[2-(3-carbamimidoyl-phenoxy)-eth...)
Affinity DataKi:  220nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127500(3,4,5,6-Tetrahydro-2H-[1,4']bipyridinyl-4-carboxyl...)
Affinity DataKi:  290nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127499(3-[4-Carbamimidoyl-2-(2-{4-[1-(1-imino-ethyl)-pipe...)
Affinity DataKi:  330nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127505(CHEMBL55364 | N-[2-(3-Carbamimidoyl-phenoxy)-ethyl...)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibitory activity against Coagulation factor X (fXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127501(3-(4-Carbamimidoyl-2-{2-[4-(pyrrolidine-1-carbonyl...)
Affinity DataKi:  2.40E+4nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127498(3-{4-Carbamimidoyl-2-[2-(4-carbamimidoyl-benzoylam...)
Affinity DataKi:  3.80E+4nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127495(3-[4-Carbamimidoyl-2-(2-{4-[1-(1-imino-ethyl)-pipe...)
Affinity DataKi:  5.30E+4nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127504(CHEMBL55770 | N-[2-(3-Carbamimidoyl-phenoxy)-ethyl...)
Affinity DataKi:  1.10E+5nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127494(3-(4-Carbamimidoyl-2-{2-[(3,4,5,6-tetrahydro-2H-[1...)
Affinity DataKi:  1.40E+5nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127496(CHEMBL51796 | N-[2-(3-Carbamimidoyl-phenoxy)-ethyl...)
Affinity DataKi:  4.40E+5nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127492(4-[5-Carbamimidoyl-2-(2-carboxy-2-oxo-ethyl)-pheno...)
Affinity DataKi:  5.40E+5nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127502(4-[5-Carbamimidoyl-2-(2-carboxy-2-oxo-ethyl)-pheno...)
Affinity DataKi:  6.80E+5nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127497(4-Carbamimidoyl-N-[2-(3-carbamimidoyl-phenoxy)-eth...)
Affinity DataKi:  7.10E+5nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127505(CHEMBL55364 | N-[2-(3-Carbamimidoyl-phenoxy)-ethyl...)
Affinity DataKi:  8.00E+5nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127500(3,4,5,6-Tetrahydro-2H-[1,4']bipyridinyl-4-carboxyl...)
Affinity DataKi:  1.00E+6nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127506(3-(4-Carbamimidoyl-benzoylamino)-4-(3-carbamimidoy...)
Affinity DataKi: >1.50E+6nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127493(3-(4-Carbamimidoyl-2-{2-[(3,4,5,6-tetrahydro-2H-[1...)
Affinity DataKi: >1.50E+6nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127503(3-(4-Carbamimidoyl-benzoylamino)-4-(3-carbamimidoy...)
Affinity DataKi: >1.50E+6nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50127499(3-[4-Carbamimidoyl-2-(2-{4-[1-(1-imino-ethyl)-pipe...)
Affinity DataKi: >1.50E+6nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50101813(CHEBI:31399 | Cilnidipine)
Affinity DataIC50:  1.10nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50101813(CHEBI:31399 | Cilnidipine)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of Voltage-dependent L-type calcium channel in rat thoracic aorta ringMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50101813(CHEBI:31399 | Cilnidipine)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of voltage-dependent L-type calcium channel in rat thoracic aorta ring assessed as effect on high K+ induced contraction by Magnus methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Taisho Pharmaceutical

US Patent
LigandPNGBDBM166423(US9073821, 550)
Affinity DataIC50:  1.60nMpH: 8.0 T: 2°CAssay Description:To assay the activity of Pseudomonas aeruginosa LpxC enzyme, LpxC was reacted with its substrate UDP-3-O-(R-3-hydroxydecanoyl)-N-acetylglucosamine an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Taisho Pharmaceutical

US Patent
LigandPNGBDBM166411(US9073821, 376)
Affinity DataIC50:  2nMpH: 8.0 T: 2°CAssay Description:To assay the activity of Pseudomonas aeruginosa LpxC enzyme, LpxC was reacted with its substrate UDP-3-O-(R-3-hydroxydecanoyl)-N-acetylglucosamine an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Taisho Pharmaceutical

US Patent
LigandPNGBDBM166426(US9073821, 557)
Affinity DataIC50:  2.30nMpH: 8.0 T: 2°CAssay Description:To assay the activity of Pseudomonas aeruginosa LpxC enzyme, LpxC was reacted with its substrate UDP-3-O-(R-3-hydroxydecanoyl)-N-acetylglucosamine an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Taisho Pharmaceutical

US Patent
LigandPNGBDBM166418(US9073821, 434)
Affinity DataIC50:  2.80nMpH: 8.0 T: 2°CAssay Description:To assay the activity of Pseudomonas aeruginosa LpxC enzyme, LpxC was reacted with its substrate UDP-3-O-(R-3-hydroxydecanoyl)-N-acetylglucosamine an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50475660(CHEMBL201566)
Affinity DataIC50:  2.80nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Taisho Pharmaceutical

US Patent
LigandPNGBDBM166415(US9073821, 405)
Affinity DataIC50:  2.90nMpH: 8.0 T: 2°CAssay Description:To assay the activity of Pseudomonas aeruginosa LpxC enzyme, LpxC was reacted with its substrate UDP-3-O-(R-3-hydroxydecanoyl)-N-acetylglucosamine an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Taisho Pharmaceutical

US Patent
LigandPNGBDBM166409(US9073821, 211)
Affinity DataIC50:  3.10nMpH: 8.0 T: 2°CAssay Description:To assay the activity of Pseudomonas aeruginosa LpxC enzyme, LpxC was reacted with its substrate UDP-3-O-(R-3-hydroxydecanoyl)-N-acetylglucosamine an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Taisho Pharmaceutical

US Patent
LigandPNGBDBM166412(US9073821, 396)
Affinity DataIC50:  3.10nMpH: 8.0 T: 2°CAssay Description:To assay the activity of Pseudomonas aeruginosa LpxC enzyme, LpxC was reacted with its substrate UDP-3-O-(R-3-hydroxydecanoyl)-N-acetylglucosamine an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Taisho Pharmaceutical

US Patent
LigandPNGBDBM166388(US9073821, 3)
Affinity DataIC50:  3.30nMpH: 8.0 T: 2°CAssay Description:To assay the activity of Pseudomonas aeruginosa LpxC enzyme, LpxC was reacted with its substrate UDP-3-O-(R-3-hydroxydecanoyl)-N-acetylglucosamine an...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetUDP-3-O-acyl-N-acetylglucosamine deacetylase(Pseudomonas aeruginosa)
Taisho Pharmaceutical

US Patent
LigandPNGBDBM166432(US9073821, 585)
Affinity DataIC50:  3.40nMpH: 8.0 T: 2°CAssay Description:To assay the activity of Pseudomonas aeruginosa LpxC enzyme, LpxC was reacted with its substrate UDP-3-O-(R-3-hydroxydecanoyl)-N-acetylglucosamine an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
Ajinomoto

Curated by ChEMBL
LigandPNGBDBM50475658(CHEMBL201984)
Affinity DataIC50:  3.70nMAssay Description:Inhibitory activity against L-type calcium channel in SD rat thoracic aorta by Magnus methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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