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Found 50 with Last Name = 'tubaro' and Initial = 'a'
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391884(CHEMBL463574)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of sheep placental COX2 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391887(CHEMBL2147422)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of sheep placental COX2 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50006805(3-(1-(4-chlorobenzyl)-3-(tert-butylthio)-5-isoprop...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of mPGES1 in IL-1beta treated human A549 cell microsomal membrane assessed as inhibition of PGE2 formation incubated for 15 mins before ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50029593(CHEMBL7162 | N-(2-(cyclohexyloxy)-4-nitrophenyl)me...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of sheep placental COX2 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391880(CHEMBL2147423)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391884(CHEMBL463574)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391890(CHEMBL2147420)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391887(CHEMBL2147422)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of mPGES1 in IL-1beta treated human A549 cell microsomal membrane assessed as inhibition of PGE2 formation incubated for 15 mins before ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50000541((+-)-1-(1-Benzo[b]thien-2-ylethyl)-1-hydroxyurea |...)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of 5-lipoxygenase in human neutrophils assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391890(CHEMBL2147420)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of sheep placental COX2 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391890(CHEMBL2147420)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of mPGES1 in IL-1beta treated human A549 cell microsomal membrane assessed as inhibition of PGE2 formation incubated for 15 mins before ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391880(CHEMBL2147423)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibition of sheep placental COX2 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391884(CHEMBL463574)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of mPGES1 in IL-1beta treated human A549 cell microsomal membrane assessed as inhibition of PGE2 formation incubated for 15 mins before ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391883(CHEMBL2147424)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of mPGES1 in IL-1beta treated human A549 cell microsomal membrane assessed as inhibition of PGE2 formation incubated for 15 mins before ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391880(CHEMBL2147423)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibition of mPGES1 in IL-1beta treated human A549 cell microsomal membrane assessed as inhibition of PGE2 formation incubated for 15 mins before ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391887(CHEMBL2147422)
Affinity DataIC50:  1.83E+4nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391886(CHEMBL2147421)
Affinity DataIC50:  1.84E+4nMAssay Description:Inhibition of 5-lipoxygenase in human neutrophils assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391886(CHEMBL2147421)
Affinity DataIC50:  1.95E+4nMAssay Description:Inhibition of mPGES1 in IL-1beta treated human A549 cell microsomal membrane assessed as inhibition of PGE2 formation incubated for 15 mins before ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391889(CHEMBL2147419)
Affinity DataIC50:  2.72E+4nMAssay Description:Inhibition of 5-lipoxygenase in human neutrophils assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391888(CHEMBL2147418)
Affinity DataIC50:  3.95E+4nMAssay Description:Inhibition of mPGES1 in IL-1beta treated human A549 cell microsomal membrane assessed as inhibition of PGE2 formation incubated for 15 mins before ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391881(CHEMBL2147415)
Affinity DataIC50:  4.14E+4nMAssay Description:Inhibition of 5-lipoxygenase in human neutrophils assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391889(CHEMBL2147419)
Affinity DataIC50:  4.20E+4nMAssay Description:Inhibition of mPGES1 in IL-1beta treated human A549 cell microsomal membrane assessed as inhibition of PGE2 formation incubated for 15 mins before ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391883(CHEMBL2147424)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of sheep placental COX2 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391881(CHEMBL2147415)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of sheep placental COX2 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391890(CHEMBL2147420)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of 5-lipoxygenase in human neutrophils assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391882(CHEMBL2147416)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of sheep placental COX2 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391887(CHEMBL2147422)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of 5-lipoxygenase in human neutrophils assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391883(CHEMBL2147424)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of 5-lipoxygenase in human neutrophils assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391883(CHEMBL2147424)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391886(CHEMBL2147421)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of sheep placental COX2 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391886(CHEMBL2147421)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391884(CHEMBL463574)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of 5-lipoxygenase in human neutrophils assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391885(CHEMBL2147417)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of 5-lipoxygenase in human neutrophils assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391888(CHEMBL2147418)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of sheep placental COX2 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391889(CHEMBL2147419)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of sheep placental COX2 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391881(CHEMBL2147415)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of mPGES1 in IL-1beta treated human A549 cell microsomal membrane assessed as inhibition of PGE2 formation incubated for 15 mins before ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391882(CHEMBL2147416)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of 5-lipoxygenase in human neutrophils assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391882(CHEMBL2147416)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of mPGES1 in IL-1beta treated human A549 cell microsomal membrane assessed as inhibition of PGE2 formation incubated for 15 mins before ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391880(CHEMBL2147423)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of 5-lipoxygenase in human neutrophils assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391885(CHEMBL2147417)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of sheep placental COX2 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E synthase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391885(CHEMBL2147417)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of mPGES1 in IL-1beta treated human A549 cell microsomal membrane assessed as inhibition of PGE2 formation incubated for 15 mins before ad...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391888(CHEMBL2147418)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of 5-lipoxygenase in human neutrophils assessed as inhibition of LTB4 productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391889(CHEMBL2147419)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391881(CHEMBL2147415)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391882(CHEMBL2147416)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391885(CHEMBL2147417)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50391888(CHEMBL2147418)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ram seminal vesicle COX1 assessed as PGE2 production by enzyme immunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50099491(2-(4-(2-(3-cyclohexyl-1-(4-cyclohexylbutyl)ureido)...)
Affinity DataEC50:  0.600nMAssay Description:Activation of PPARalpha transfected in HEK293 cells after 18 hrs by firefly luciferase reporter gene-based luminescence assay relative to controlMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50085045(5-((4-((6-hydroxy-2,5,7,8-tetramethyl-3,4-dihydro-...)
Affinity DataEC50:  400nMAssay Description:Activation of PPARgamma transfected in HEK293 cells after 18 hrs by firefly luciferase reporter gene-based luminescence assay relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed