TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: >0.0480nMAssay Description:Binding affinity to human adenosine A2a receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 2.10nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.20nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Competitive inhibition of human neutrophil elastase using N-methylsuccinyl-Ala-Ala-Pro-Val-7-amino-4-methylcoumarin as substrate by Dixon plot analys...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity to bovine adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Binding affinity to human adenosine A2b receptorMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 35nMAssay Description:Inhibition of human neutrophil elastaseMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2b(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2b receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Competitive inhibition of human neutrophil elastase using N-methylsuccinyl-Ala-Ala-Pro-Val-7-amino-4-methylcoumarin as substrate by Dixon plot analys...More data for this Ligand-Target Pair
TargetAdenosine receptor A3(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 64nMAssay Description:Displacement of [125I]AB-MECA from human adenosine A3 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 68nMAssay Description:Binding affinity to human adenosine A2a receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 69nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Dipartimento Di Scienze Farmaceutiche
Curated by ChEMBL
Affinity DataKi: 76nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 85nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 93nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 104nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 123nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 173nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Binding affinity to human adenosine A1 receptorMore data for this Ligand-Target Pair