Affinity DataKi: 8.90nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 13.3nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 17.9nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 30.4nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 69.2nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 76.6nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 89.4nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 95.3nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 241nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 241nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 284nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 325nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 335nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 344nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 349nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 533nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 534nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 561nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 605nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 678nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB1 receptor in rat brain membrane in presence of phenylmethanesulfonyl fluorideMore data for this Ligand-Target Pair
Affinity DataKi: 750nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 826nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 840nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 868nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 869nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 987nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.03E+3nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.05E+3nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.12E+3nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.56E+3nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.04E+3nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 3.26E+3nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Displacement of [3H]CP55940 from cannabinoid CB2 receptor in mouse spleen membraneMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of electric eel acetylcholinesterase using acetylthiocholine as substrate incubated for 15 mins followed by substrate addition measured fo...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Inhibition of electric eel acetylcholinesterase using acetylthiocholine as substrate incubated for 15 mins followed by substrate addition measured fo...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Inhibition of electric eel acetylcholinesterase using acetylthiocholine as substrate incubated for 15 mins followed by substrate addition measured fo...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Inhibition of electric eel acetylcholinesterase using acetylthiocholine as substrate incubated for 15 mins followed by substrate addition measured fo...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 3.10nMAssay Description:Inhibition of electric eel acetylcholinesterase using acetylthiocholine as substrate incubated for 15 mins followed by substrate addition measured fo...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 3.90nMAssay Description:Inhibition of electric eel acetylcholinesterase using acetylthiocholine as substrate incubated for 15 mins followed by substrate addition measured fo...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of electric eel acetylcholinesterase using acetylthiocholine as substrate incubated for 15 mins followed by substrate addition measured fo...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 9.30nMAssay Description:Inhibition of electric eel acetylcholinesterase using acetylthiocholine as substrate incubated for 15 mins followed by substrate addition measured fo...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of electric eel acetylcholinesterase using acetylthiocholine as substrate incubated for 15 mins followed by substrate addition measured fo...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of electric eel acetylcholinesterase using acetylthiocholine as substrate incubated for 15 mins followed by substrate addition measured fo...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of electric eel acetylcholinesterase using acetylthiocholine as substrate incubated for 15 mins followed by substrate addition measured fo...More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of horse serum butyrylcholinesterase using butylthiocholine as substrate incubated for 15 mins followed by substrate addition measured for...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Sun Yat-Sen University
Curated by ChEMBL
Sun Yat-Sen University
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Inhibition of electric eel acetylcholinesterase using acetylthiocholine as substrate incubated for 15 mins followed by substrate addition measured fo...More data for this Ligand-Target Pair