Affinity DataKi: 0.640nMAssay Description:Displacement of [125I]SS-14 from human SST3 receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity to human SST3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of human CA9 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Inhibition of human CA2 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Inhibition of human CA9 preincubated for 15 mins prior to testing by phenol red-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Inhibition of human CA9 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Inhibition of human CA12 preincubated for 15 mins prior to testing by phenol red-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Inhibition of human CA12 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of recombinant human carbonic anhydrase 12 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Inhibition of human CA12 preincubated for 15 mins prior to testing by phenol red-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Inhibition of human CA9 preincubated for 15 mins prior to testing by phenol red-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Inhibition of human CA9 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.20nMAssay Description:Inhibition of human CA12 preincubated for 15 mins prior to testing by phenol red-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:Inhibition of human CA9 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of human CA2 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.10nMAssay Description:Inhibition of human CA12 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.40nMAssay Description:Inhibition of human CA9 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University Of Kansas
Curated by PDSP Ki Database
University Of Kansas
Curated by PDSP Ki Database
Affinity DataKi: 9.60nMAssay Description:Inhibition of human CA12 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Inhibition of human CA2 preincubated for 15 mins prior to testing by phenol red-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:Inhibition of human CA9 preincubated for 15 mins prior to testing by phenol red-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:Inhibition of human CA2 preincubated for 15 mins prior to testing by phenol red-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of human CA9 preincubated for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of recombinant human carbonic anhydrase 2 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of human CA9 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of human CA12 preincubated for 15 mins prior to testing by phenol red-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of human CA2 preincubated for 15 mins prior to testing by phenol red-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of human CA9 preincubated for 15 mins prior to testing by phenol red-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University Of Kansas
Curated by PDSP Ki Database
University Of Kansas
Curated by PDSP Ki Database
Affinity DataKi: 12nMAssay Description:Inhibition of human CA2 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of human CA2 preincubated for 15 mins prior to testing by phenol red-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of human CA9 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Inhibition of recombinant full length stromelysin (FLS)More data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Inhibition of human CA12 preincubated for 15 mins prior to testing by phenol red-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of recombinant stromelysin catalytic domain (SCD)More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of human CA2 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of human CA12 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University Of Kansas
Curated by PDSP Ki Database
University Of Kansas
Curated by PDSP Ki Database
Affinity DataKi: 17nMAssay Description:Inhibition of human CA12 preincubated for 15 mins prior to testing by phenol red-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of human CA12 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chongqing Medical University
Curated by ChEMBL
Chongqing Medical University
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Binding affinity to GST-tagged PPARG LBD (unknown origin) by Fluormone Pan-PPAR Green tracer based TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of human CA12 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: <17.7nMAssay Description:Inhibition of Staphylococcus aureus DNA gyraseMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibition of human CA2 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Inhibition of human CA12 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of human CA9 by stopped- flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of recombinant human carbonic anhydrase 9 preincubated with enzyme for 15 mins by phenol red dye based stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Inhibition of human CA9 preincubated for 15 mins prior to testing by phenol red-based stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University Of Kansas
Curated by PDSP Ki Database
University Of Kansas
Curated by PDSP Ki Database
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University Of Kansas
Curated by PDSP Ki Database
University Of Kansas
Curated by PDSP Ki Database