Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 87 hits for monomerid = 50072864,50072865,50072861,50073910,50073915,50073918,50073912,50073909,50073913,50073914,50087245,50085865,50093125,50099447,50099448,50099449,50099450,50099451,50099452,50102025,50102026,50118686,50118687,50122792,50122793,50122795,50122796,50122797,50129630,50129631,50129632,50129633,50129634,50139762,50139763,50139764,50143944,50161189,50168313,50168314,50168317,50168318,50168312,50193152,50208564,50208565,50208566,50208568,50208569,50208570,50208571,50336688   

TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50102025(4-[(10S,14S,18S)-18-(2-AMINO-2-OXOETHYL)-14-(1-NAP...)
Affinity DataKi:  16nMAssay Description:Displacement of FITC-Ahx-PVPePYINQSVPKRK-NH2 from N-terminal His6-tagged human full length GRB2 (1 to 217 residues) expressed in Escherichia coli ass...More data for this Ligand-Target Pair
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50118686(CHEMBL323505 | [(S)-3-(2-Azido-2-{1-[(S)-2-carbamo...)
Affinity DataIC50: >3.00E+4nMAssay Description:Binding affinity for Growth factor receptor bound protein 2 SH2 domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50118687((R)-N-{1-[(S)-2-Carbamoyl-1-(3-naphthalen-1-yl-pro...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain binding to p185erbB-2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50072865(CHEMBL55627 | N-[(S)-1-{1-[(S)-2-Carbamoyl-1-(3-na...)
Affinity DataIC50:  9nMAssay Description:Binding affinity for Growth factor receptor bound protein 2 SH2 domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50072864(CHEMBL115699 | {[4-((S)-2-Acetylamino-2-{1-[(S)-2-...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Grb2 SH2 domain binding in MDA-MB-453 human breast carcinoma cell lysatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50072861(CHEMBL19417 | [(S)-4-(2-Acetylamino-2-{1-[2-carbam...)
Affinity DataIC50:  80nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain binding in plasmon resonance binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50073909(CHEMBL72036 | {4-[(S)-2-Acetylamino-2-(1-{(S)-2-ca...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of Grb-SH2 domain binding to phosphorylated carboxy-terminal intracellular domain of epidermal growth factor receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50073910(CHEMBL431381 | {4-[(S)-2-Acetylamino-2-(1-{(S)-2-c...)
Affinity DataIC50:  59nMAssay Description:Inhibition of Grb-SH2 domain binding to phosphorylated carboxy-terminal intracellular domain of epidermal growth factor receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50073913(CHEMBL73003 | {4-[(S)-2-Acetylamino-2-(1-{(S)-2-ca...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of Grb-SH2 domain binding to phosphorylated carboxy-terminal intracellular domain of epidermal growth factor receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50073912(CHEMBL72996 | {4-[(S)-2-Acetylamino-2-(1-{(S)-2-ca...)
Affinity DataIC50:  9.20nMAssay Description:Inhibition of Grb-SH2 domain binding to phosphorylated carboxy-terminal intracellular domain of epidermal growth factor receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50073915(CHEMBL72114 | {4-[(S)-2-Acetylamino-2-(1-{(S)-2-ca...)
Affinity DataIC50:  81nMAssay Description:Inhibition of Grb-SH2 domain binding to phosphorylated carboxy-terminal intracellular domain of epidermal growth factor receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50073914(CHEMBL71034 | {4-[(S)-2-Acetylamino-2-(1-{(S)-2-ca...)
Affinity DataIC50:  155nMAssay Description:Inhibition of Grb-SH2 domain binding to phosphorylated carboxy-terminal intracellular domain of epidermal growth factor receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50073918(CHEMBL431982 | [4-((S)-2-Acetylamino-2-{1-[(S)-2-c...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of Grb-SH2 domain binding to phosphorylated carboxy-terminal intracellular domain of epidermal growth factor receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50072861(CHEMBL19417 | [(S)-4-(2-Acetylamino-2-{1-[2-carbam...)
Affinity DataIC50:  80nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain binding in plasmon resonance binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50072865(CHEMBL55627 | N-[(S)-1-{1-[(S)-2-Carbamoyl-1-(3-na...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Grb2 SH2 domain binding in MDA-MB-453 human breast carcinoma cell lysatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50072864(CHEMBL115699 | {[4-((S)-2-Acetylamino-2-{1-[(S)-2-...)
Affinity DataIC50:  80nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain binding in plasmon resonance binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50087245(CHEMBL345170 | Pro-Ser-Pmp-Val-Asn-Val-Gln-Asn)
Affinity DataKd:  260nMAssay Description:Dissociation constant of compound was determined from affinity of compound towards Growth factor receptor bound protein 2 measured by fluorescenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50085865(2-[4-(2-Acetylamino-2-{1-[2-carbamoyl-1-(3-naphtha...)
Affinity DataIC50:  160nMAssay Description:Inhibition of Growth factor receptor bound protein 2 binding by ELISA assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50072865(CHEMBL55627 | N-[(S)-1-{1-[(S)-2-Carbamoyl-1-(3-na...)
Affinity DataIC50:  50nMAssay Description:Inhibition of Growth factor receptor bound protein 2 binding by ELISA assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50073909(CHEMBL72036 | {4-[(S)-2-Acetylamino-2-(1-{(S)-2-ca...)
Affinity DataIC50:  4nMAssay Description:Inhibition of Growth factor receptor bound protein 2 binding by ELISA assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50072861(CHEMBL19417 | [(S)-4-(2-Acetylamino-2-{1-[2-carbam...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Growth factor receptor bound protein 2 binding by ELISA assay methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50093125((4-{(S)-2-Acetylamino-2-[1-((1R,2S)-2-carbamoyl-cy...)
Affinity DataIC50:  700nMAssay Description:Inhibition of Grb2-SH2 domain binding to phospho-EGF receptor intracellular C-terminal domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50099448(CHEMBL276300 | {4-[(S)-2-Acetylamino-2-(1-{(S)-2-c...)
Affinity DataIC50:  25nMAssay Description:Inhibitory concentration required against Src homology (SH2) domain of Growth factor receptor bound protein 2 by ELISA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50099447(CHEMBL278567 | {4-[(S)-2-Acetylamino-2-(1-{(S)-2-c...)
Affinity DataIC50:  43nMAssay Description:Inhibitory concentration required against Src homology (SH2) domain of Growth factor receptor bound protein 2 by ELISA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50099449(CHEMBL281577 | {4-[(S)-2-Acetylamino-2-(1-{(S)-2-c...)
Affinity DataIC50:  130nMAssay Description:Inhibitory concentration required against Src homology (SH2) domain of Growth factor receptor bound protein 2 by ELISA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50072861(CHEMBL19417 | [(S)-4-(2-Acetylamino-2-{1-[2-carbam...)
Affinity DataIC50:  43nMAssay Description:Inhibitory concentration required against Src homology (SH2) domain of Growth factor receptor bound protein 2 by ELISA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50099450(CHEMBL19378 | {4-[(S)-2-Acetylamino-2-(1-{(S)-2-ca...)
Affinity DataIC50:  11nMAssay Description:Inhibitory concentration required against Src homology (SH2) domain of Growth factor receptor bound protein 2 by ELISA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50099452(CGP-78850 | CHEMBL276046 | {4-[(S)-2-Acetylamino-2...)
Affinity DataIC50:  43nMAssay Description:Inhibitory concentration required against Src homology (SH2) domain of Growth factor receptor bound protein 2 by ELISA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50099451(CHEMBL19214 | {4-[(S)-2-Acetylamino-2-(1-{(S)-2-ca...)
Affinity DataIC50:  84nMAssay Description:Inhibitory concentration required against Src homology (SH2) domain of Growth factor receptor bound protein 2 by ELISA binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50102025(4-[(10S,14S,18S)-18-(2-AMINO-2-OXOETHYL)-14-(1-NAP...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain binding in ELISAMore data for this Ligand-Target Pair
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50102026(CHEMBL292883 | [4-(2-{1-[2-Carbamoyl-1-(3-naphthal...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain binding in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50072865(CHEMBL55627 | N-[(S)-1-{1-[(S)-2-Carbamoyl-1-(3-na...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain binding in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50072861(CHEMBL19417 | [(S)-4-(2-Acetylamino-2-{1-[2-carbam...)
Affinity DataIC50:  55nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain binding in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50139762(CHEMBL349373 | [(16R,20S)-18-((S)-Carbamoylmethyl)...)
Affinity DataKd:  0.0750nMAssay Description:Binding affinity to SH2 domain of GRB2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50139762(CHEMBL349373 | [(16R,20S)-18-((S)-Carbamoylmethyl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SH2 domain of GRB2 in human MDA-MB-231 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50122793(CHEMBL313407 | {4-[3-Carbamoylmethyl-14-(2,3-dihyd...)
Affinity DataIC50:  700nMAssay Description:Inhibition against Growth factor receptor bound protein 2 binding using ELISA techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50122795(CHEMBL315337 | [4-(19-Carbamoylmethyl-15-naphthale...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition against Growth factor receptor bound protein 2 binding using ELISA techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50122796(CHEMBL84798 | [18-Carbamoylmethyl-14-(2,3-dihydro-...)
Affinity DataIC50:  2nMAssay Description:Inhibition against Growth factor receptor bound protein 2 binding using ELISA techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50122792(CHEMBL312875 | [3-Carbamoylmethyl-14-(2,3-dihydro-...)
Affinity DataIC50:  8nMAssay Description:Inhibition against Growth factor receptor bound protein 2 binding using ELISA techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50122797(CHEMBL406148 | i{4-[18-Carbamoylmethyl-14-(2,3-dih...)
Affinity DataIC50:  20nMAssay Description:Inhibition against Growth factor receptor bound protein 2 binding using ELISA techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50129630(CHEMBL422957 | [4-(18-Carbamoylmethyl-8,12,17,20-t...)
Affinity DataIC50:  4.79E+4nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain in extracellular binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50129631((4-{2-[1-(1,2-Dicarbamoyl-ethylcarbamoyl)-cyclohex...)
Affinity DataIC50:  5.25E+4nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain in extracellular binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50129632(CHEMBL91584 | [4-(16-Carbamoylmethyl-8,12,15,18-te...)
Affinity DataIC50: >6.00E+5nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain in extracellular binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50102025(4-[(10S,14S,18S)-18-(2-AMINO-2-OXOETHYL)-14-(1-NAP...)
Affinity DataIC50:  26nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain in extracellular binding assayMore data for this Ligand-Target Pair
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50129633(CHEMBL91880 | [4-(17-Carbamoylmethyl-8,12,16,19-te...)
Affinity DataIC50: >6.00E+5nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain in extracellular binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50129634(CHEMBL90990 | [4-(18-Carbamoylmethyl-14-naphthalen...)
Affinity DataIC50:  7.90E+3nMAssay Description:Inhibition of Growth factor receptor bound protein 2 SH2 domain in extracellular binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50139762(CHEMBL349373 | [(16R,20S)-18-((S)-Carbamoylmethyl)...)
Affinity DataKd:  0.0930nMAssay Description:In vitro binding affinity for Grb2 SH2 domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50102025(4-[(10S,14S,18S)-18-(2-AMINO-2-OXOETHYL)-14-(1-NAP...)
Affinity DataIC50:  20nMAssay Description:In vitro binding affinity in extracellular ELISA-based assay for Grb2 SH2 domainMore data for this Ligand-Target Pair
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50139763(CHEMBL306657 | [(E)-(9S,10S,14S,18S)-18-Carbamoylm...)
Affinity DataIC50:  2nMAssay Description:In vitro binding affinity in extracellular ELISA-based assay for Grb2 SH2 domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGrowth factor receptor-bound protein 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50139764(5-Methylindolyl derivative | CHEMBL423988)
Affinity DataKd:  0.0750nMAssay Description:In vitro binding affinity for Grb2 SH2 domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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