Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 63 hits for monomerid = 50104296,50163440,50182798,50288855,50150471,50235814,50235812,50235815
TargetAlpha-galactosidase(Coffea arabica (Coffee beans))
Technische Universit£T Graz
Curated by ChEMBL
Technische Universit£T Graz
Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Inhibition of alpha-galactosidase green coffee beansMore data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Inhibition of Escherichia coli lacZ beta-galactosidase using 4-nitrophenyl-beta-D-galactopyranoside as substrate preincubated up to 5 mins followed b...More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Technical University Graz
Curated by ChEMBL
Technical University Graz
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Inhibition of human lysosomal beta-glucocerebrosidaseMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Technical University Graz
Curated by ChEMBL
Technical University Graz
Curated by ChEMBL
Affinity DataKi: 2.80E+3nMpH: 5.0Assay Description:Competitive inhibition of wild type human glucocerebrosidase using 2,4-dinitrophenyl beta-D-glucopyranoside as substrate after 3 mins by Dixon and Li...More data for this Ligand-Target Pair
Affinity DataKi: 4.00E+3nMAssay Description:Inhibition of bovine liver beta-galactosidase using 4-nitrophenyl-beta-D-galactopyranoside as substrate preincubated up to 5 mins followed by substra...More data for this Ligand-Target Pair
Affinity DataKi: 1.25E+4nMAssay Description:Inhibition of Agrobacterium sp. beta-galactosidaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+4nMAssay Description:Inhibitory activity towards Beta-galactosidase from Jack beanMore data for this Ligand-Target Pair
Affinity DataKi: 2.70E+4nMAssay Description:Inhibitory activity towards Beta-Glucosidase from AlmondMore data for this Ligand-Target Pair
TargetBeta-glucosidase A(Caldocellum saccharolyticum)
Section De Chimie De L'Universit£
Curated by ChEMBL
Section De Chimie De L'Universit£
Curated by ChEMBL
Affinity DataKi: 2.70E+4nMAssay Description:Inhibitory activity towards Beta-Glucosidase from Caldocellum saccharolMore data for this Ligand-Target Pair
Affinity DataKi: 4.47E+4nM ΔG°: -6.17kcal/molepH: 4.5 T: 2°CAssay Description:β-Gal activity was measured by using 4-methylumbelliferyll-β-D-galactopyranoside in buffer B (0.15 M sodium citrate, pH 4.5, and 0.2 M NaCl...More data for this Ligand-Target Pair
Affinity DataKi: 4.90E+4nM ΔG°: -6.11kcal/molepH: 4.5 T: 2°CAssay Description:β-Gal activity was measured by using 4-methylumbelliferyll-β-D-galactopyranoside in buffer B (0.15 M sodium citrate, pH 4.5, and 0.2 M NaCl...More data for this Ligand-Target Pair
Affinity DataKi: 5.00E+4nMAssay Description:Inhibition of Agrobacterium sp. beta glucosidaseMore data for this Ligand-Target Pair
Affinity DataKi: 6.18E+4nM ΔG°: -5.97kcal/molepH: 4.5 T: 2°CAssay Description:β-Gal activity was measured by using 4-methylumbelliferyll-β-D-galactopyranoside in buffer B (0.15 M sodium citrate, pH 4.5, and 0.2 M NaCl...More data for this Ligand-Target Pair
Affinity DataKi: 8.00E+4nMAssay Description:Inhibitory activity towards Alpha-mannosidase from Jack beanMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+5nMAssay Description:Inhibitory activity towards Beta-galactosidase from Aspergillus nigerMore data for this Ligand-Target Pair
TargetBeta-xylosidase(Thermoanaerobacter saccharolyticum)
Technische UniversitäT Graz
Curated by ChEMBL
Technische UniversitäT Graz
Curated by ChEMBL
Affinity DataKi: 2.06E+5nMAssay Description:Inhibition of Thermoanaerobacterium saccharolyticum beta-xylosidaseMore data for this Ligand-Target Pair
Affinity DataKi: >2.00E+6nMAssay Description:Inhibition of human recombinant lysosomal alpha-galactosidase using 2,4-dinitrophenyl-alpha-D-galactopyranoside as substrate preincubated up to 5 min...More data for this Ligand-Target Pair
Affinity DataKi: 3.40E+7nMAssay Description:Inhibition constant against Alpha-FucosidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of lysosomal alpha-glucosidase by HPLCMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Technical University Graz
Curated by ChEMBL
Technical University Graz
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human GCaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of maltase by HPLCMore data for this Ligand-Target Pair
TargetBeta-glucosidase A(Caldocellum saccharolyticum)
Section De Chimie De L'Universit£
Curated by ChEMBL
Section De Chimie De L'Universit£
Curated by ChEMBL
Affinity DataIC50: 3.67E+5nMpH: 5.0Assay Description:Inhibition of Caldocellum saccharolyticum beta-glucosidase assessed as p-nitrophenol release at pH 5 by spectrometric analysisMore data for this Ligand-Target Pair
TargetAlpha-galactosidase(Coffea arabica (Coffee beans))
Technische Universit£T Graz
Curated by ChEMBL
Technische Universit£T Graz
Curated by ChEMBL
Affinity DataIC50: 3nMpH: 6.5Assay Description:Inhibition of coffee bean alpha-galactosidase assessed as p-nitrophenol release at pH 6.5 by spectrometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of human lysosome alpha-galactosidase assessed as p-nitrophenol release by spectrometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 7.20E+4nMAssay Description:Inhibition of rat intestinal lactase assessed as p-nitrophenol release by spectrometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+5nMAssay Description:Inhibitory activity towards Beta-galactosidase from Jack beanMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibitory concentration against human alpha-galactosidaseMore data for this Ligand-Target Pair
TargetAlpha-galactosidase C(Aspergillus niger)
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibitory concentration against alpha-galactosidase of Aspergillus nigerMore data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibitory concentration against human beta-galactosidaseMore data for this Ligand-Target Pair
TargetBeta-galactosidase(Rattus norvegicus)
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Toyama Medical And Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibitory concentration against beta-galactosidase of ratMore data for this Ligand-Target Pair
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibitory activity towards Alpha-mannosidase from Jack beanMore data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Technical University Graz
Curated by ChEMBL
Technical University Graz
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human lysosomal beta-glucosidaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+5nMAssay Description:Inhibitory activity towards Alpha-mannosidase from Jack beanMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40E+5nMAssay Description:Inhibitory activity towards Beta-galactosidase from Aspergillus nigerMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human alpha GAL-A using 4-methylumbelliferyl alpha-D-galactopyranoside as substrate at pH 7 after 15 mins by fluorescence a...More data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of recombinant human alpha GAL-A using 4-methylumbelliferyl alpha-D-galactopyranoside as substrate at pH 4.6 after 15 mins by fluorescence...More data for this Ligand-Target Pair
Affinity DataIC50: >1.60E+5nMAssay Description:Inhibitory concentration against cyclin dependent kinase-2 (CDK2)/Cyclin EMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibitory concentration against cyclin dependent kinase-2 (CDK2)/Cyclin EMore data for this Ligand-Target Pair
Affinity DataIC50: >1.50E+5nMAssay Description:Inhibitory concentration against cyclin dependent kinase-2 (CDK2)/Cyclin EMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibitory concentration against cyclin dependent kinase-2 (CDK2)/Cyclin EMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibitory concentration against cyclin dependent kinase-2 (CDK2)/Cyclin EMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of alpha-glucosidase derived from human peripheral blood mononuclear cell lysate using 4-methylumbelliferyl alpha-D-glucopyranoside as sub...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of beta-galactosidase derived from human peripheral blood mononuclear cell lysate using 4-methylumbelliferyl beta-D-galactopyranoside as s...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of beta-glucosidase derived from human peripheral blood mononuclear cell lysate using 4-methylumbelliferyl beta-D-glucopyranoside as subst...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of GBA2 by HPLCMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of lactase by HPLCMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GCS by cell-based assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.30E+4nMAssay Description:Compound was evaluated for inhibition of beta-galactosidase from aspergillus oryzae (sigma G 7256).More data for this Ligand-Target Pair
TargetLysosomal acid glucosylceramidase(Homo sapiens (Human))
Technical University Graz
Curated by ChEMBL
Technical University Graz
Curated by ChEMBL
Affinity DataIC50: 5.30E+5nMAssay Description:Compound was evaluated for inhibition of beta-glucosidase from almonds(sigma G 4511).More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+6nMAssay Description:Compound was evaluated for inhibition of alpha-fucosidase from bovine kidney(sigma F 5884).More data for this Ligand-Target Pair
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