Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50441972,50441973,50441974,50441975,50441976,50441977   

TargetCytohesin-2(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50441975(CHEMBL2440216)
Affinity DataKi:  5.40E+5nMAssay Description:Inhibition of human Arno Sec7 domain-mediated nucleotide exchange in delta17 Arf1 (17 to 181) by BODIPY-GTP based time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytohesin-2(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50441972(CHEMBL2440207)
Affinity DataKi:  9.80E+5nMAssay Description:Inhibition of human Arno Sec7 domain-mediated nucleotide exchange in delta17 Arf1 (17 to 181) by BODIPY-GTP based time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytohesin-2(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50441973(CHEMBL2440218)
Affinity DataKi:  1.61E+6nMAssay Description:Inhibition of human Arno Sec7 domain-mediated nucleotide exchange in delta17 Arf1 (17 to 181) by BODIPY-GTP based time resolved fluorescence assayMore data for this Ligand-Target Pair
TargetCytohesin-2(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50441976(CHEMBL2440213)
Affinity DataKi:  1.91E+6nMAssay Description:Inhibition of human Arno Sec7 domain-mediated nucleotide exchange in delta17 Arf1 (17 to 181) by BODIPY-GTP based time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytohesin-2(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50441977(CHEMBL2440208)
Affinity DataKi:  3.72E+6nMAssay Description:Inhibition of human Arno Sec7 domain-mediated nucleotide exchange in delta17 Arf1 (17 to 181) by BODIPY-GTP based time resolved fluorescence assayMore data for this Ligand-Target Pair
TargetCytohesin-2(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50441974(CHEMBL236358)
Affinity DataKi:  5.12E+6nMAssay Description:Inhibition of human Arno Sec7 domain-mediated nucleotide exchange in delta17 Arf1 (17 to 181) by BODIPY-GTP based time resolved fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50441973(CHEMBL2440218)
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human FFA4 receptor expressed in U2OS cells assessed as calcium mobilization after 24 hrs by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytohesin-2(Homo sapiens (Human))
University Of Montpellier

Curated by ChEMBL
LigandPNGBDBM50441977(CHEMBL2440208)
Affinity DataKd:  5.00E+5nMAssay Description:Binding affinity to human Arno Sec7 domain immobilized on CAP sensor chip after 15 mins by 1H 1D-NMR-700 MHz spectra analysisMore data for this Ligand-Target Pair