Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 62 hits for monomerid = 6676,6677,6678,6679,6680,6681,6682,6683,6684,6685,6686,6687,6688,6689,6690,6691,6692,6693,6694,6695,6696,6697,6699,6700,6701,6702,6703,6704,6705   

TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6676(3-benzoyl-6-[(2,6-difluorophenyl)carbonyl]imidazo[...)
Affinity DataIC50:  324nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM6683(aminoimidazo[1,2-a]pyridine deriv. 18 | {2-amino-6...)
Affinity DataIC50:  105nMAssay Description:Inhibition of recombinant human CDK1/cyclin B expressed in baculovirus infected Sf9 insect cells using histone H1 as substrate in presence of [gamma3...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6678(3-[(2-chloro-6-fluorophenyl)carbonyl]-6-[(2,6-difl...)
Affinity DataIC50:  102nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6679(3-[(2,6-difluoro-4-methoxyphenyl)carbonyl]-6-[(2,6...)
Affinity DataIC50:  91nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6680(6-[(2,6-difluorophenyl)carbonyl]-3-[(2-methoxyphen...)
Affinity DataIC50:  68nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6681(3-[(2,6-dichlorophenyl)carbonyl]-6-[(2,6-difluorop...)
Affinity DataIC50:  121nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6682(aminoimidazo[1,2-a]pyridine deriv. 17 | {2-amino-6...)
Affinity DataIC50:  214nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6683(aminoimidazo[1,2-a]pyridine deriv. 18 | {2-amino-6...)
Affinity DataIC50:  26nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6684(aminoimidazo[1,2-a]pyridine deriv. 20 | {2-amino-6...)
Affinity DataIC50:  29nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6685(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50:  95nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6686(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50:  46nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6687(6-[(2-chloro-6-fluorophenyl)carbonyl]-3-[(2,6-difl...)
Affinity DataIC50:  33nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6688(3-[(2,6-difluorophenyl)carbonyl]-6-[1-(2,6-difluor...)
Affinity DataIC50:  63nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6689((2E)-3-{2-amino-3-[(2,6-difluorophenyl)carbonyl]im...)
Affinity DataIC50:  160nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6690(6-[(Z)-1-(2,6-difluorophenyl)-2-(1H-1,2,3,4-tetraz...)
Affinity DataIC50:  1.69E+3nMpH: 7.0 T: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM6676(3-benzoyl-6-[(2,6-difluorophenyl)carbonyl]imidazo[...)
Affinity DataIC50:  326nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM6677(3,6-bis[(2,6-difluorophenyl)carbonyl]imidazo[1,2-a...)
Affinity DataIC50:  57nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM6687(6-[(2-chloro-6-fluorophenyl)carbonyl]-3-[(2,6-difl...)
Affinity DataIC50:  104nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM6688(3-[(2,6-difluorophenyl)carbonyl]-6-[1-(2,6-difluor...)
Affinity DataIC50:  93nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM6689((2E)-3-{2-amino-3-[(2,6-difluorophenyl)carbonyl]im...)
Affinity DataIC50:  53nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM6690(6-[(Z)-1-(2,6-difluorophenyl)-2-(1H-1,2,3,4-tetraz...)
Affinity DataIC50:  96nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM6680(6-[(2,6-difluorophenyl)carbonyl]-3-[(2-methoxyphen...)
Affinity DataIC50:  475nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM6681(3-[(2,6-dichlorophenyl)carbonyl]-6-[(2,6-difluorop...)
Affinity DataIC50:  209nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM6678(3-[(2-chloro-6-fluorophenyl)carbonyl]-6-[(2,6-difl...)
Affinity DataIC50:  239nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM6679(3-[(2,6-difluoro-4-methoxyphenyl)carbonyl]-6-[(2,6...)
Affinity DataIC50:  132nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM6682(aminoimidazo[1,2-a]pyridine deriv. 17 | {2-amino-6...)
Affinity DataIC50:  165nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM6683(aminoimidazo[1,2-a]pyridine deriv. 18 | {2-amino-6...)
Affinity DataIC50:  105nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM6684(aminoimidazo[1,2-a]pyridine deriv. 20 | {2-amino-6...)
Affinity DataIC50:  143nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM6685(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50:  328nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia Cancer Research Institute

Curated by ChEMBL
LigandPNGBDBM6686(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50:  154nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6676(3-benzoyl-6-[(2,6-difluorophenyl)carbonyl]imidazo[...)
Affinity DataIC50:  5.05E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6677(3,6-bis[(2,6-difluorophenyl)carbonyl]imidazo[1,2-a...)
Affinity DataIC50:  1.08E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6687(6-[(2-chloro-6-fluorophenyl)carbonyl]-3-[(2,6-difl...)
Affinity DataIC50:  810nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6688(3-[(2,6-difluorophenyl)carbonyl]-6-[1-(2,6-difluor...)
Affinity DataIC50:  1.03E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6689((2E)-3-{2-amino-3-[(2,6-difluorophenyl)carbonyl]im...)
Affinity DataIC50:  1.55E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6690(6-[(Z)-1-(2,6-difluorophenyl)-2-(1H-1,2,3,4-tetraz...)
Affinity DataIC50:  1.70E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6680(6-[(2,6-difluorophenyl)carbonyl]-3-[(2-methoxyphen...)
Affinity DataIC50:  1.97E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6681(3-[(2,6-dichlorophenyl)carbonyl]-6-[(2,6-difluorop...)
Affinity DataIC50:  359nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6678(3-[(2-chloro-6-fluorophenyl)carbonyl]-6-[(2,6-difl...)
Affinity DataIC50:  827nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6679(3-[(2,6-difluoro-4-methoxyphenyl)carbonyl]-6-[(2,6...)
Affinity DataIC50:  838nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6682(aminoimidazo[1,2-a]pyridine deriv. 17 | {2-amino-6...)
Affinity DataIC50:  1.89E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6683(aminoimidazo[1,2-a]pyridine deriv. 18 | {2-amino-6...)
Affinity DataIC50:  786nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6684(aminoimidazo[1,2-a]pyridine deriv. 20 | {2-amino-6...)
Affinity DataIC50:  464nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6685(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50:  2.59E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6686(4-({2-amino-6-[(2,6-dichlorophenyl)carbonyl]imidaz...)
Affinity DataIC50:  1.14E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6691(6-benzoyl-3-[(2,6-difluorophenyl)carbonyl]imidazo[...)
Affinity DataIC50:  1.93E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6692(6-[(2-chlorophenyl)carbonyl]-3-[(2,6-difluoropheny...)
Affinity DataIC50:  428nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6693(3-[(2,6-difluorophenyl)carbonyl]-6-{[2-(trifluorom...)
Affinity DataIC50:  1.07E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6694(3-[(2,6-difluorophenyl)carbonyl]-6-[(2-methylpheny...)
Affinity DataIC50:  1.29E+3nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Avenida De La Industria

LigandPNGBDBM6695(3-[(2,6-difluorophenyl)carbonyl]-6-[(2-methoxyphen...)
Affinity DataIC50:  603nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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