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Found 18 Enz. Inhib. hit(s) with Target = 'Chromobox protein homolog 6'
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50538817(CHEMBL4646032)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of CBX6 (unknown origin) assessed as inhibition of CBX4 disruption by competitive FP assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50538816(CHEMBL4642464)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of CBX6 (unknown origin) assessed as inhibition of CBX4 disruption by competitive FP assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50538815(CHEMBL4640937)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of CBX6 (unknown origin) assessed as inhibition of CBX4 disruption by competitive FP assayMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50157430(CHEMBL3781271)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of CBX6 (unknown origin) assessed as inhibition of CBX4 disruption by competitive FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50194259(CHEMBL3939958)
Affinity DataKd:  610nMAssay Description:Binding affinity to human N-terminal his-tagged CBX6 chromodomain (8 to 65 residues) expressed in Escherichia coli Rosetta BL21(DE3)pLysS by ITC meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50538808(CHEMBL4646516)
Affinity DataKd:  900nMAssay Description:Binding affinity to CBX6 (unknown origin) assessed as dissociation constant by fluorescence polarization analysisMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50538809(CHEMBL4637043)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to CBX6 (unknown origin) assessed as dissociation constant by fluorescence polarization analysisMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50538810(CHEMBL4647581)
Affinity DataKd:  78nMAssay Description:Binding affinity to CBX6 (unknown origin) assessed as dissociation constant by fluorescence polarization analysisMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50155931(CHEMBL3780251)
Affinity DataKd:  47nMAssay Description:Binding affinity to CBX6 (unknown origin) assessed as dissociation constant by fluorescence polarization analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50538811(CHEMBL4640223)
Affinity DataKd:  800nMAssay Description:Binding affinity to CBX6 (unknown origin) assessed as dissociation constant by fluorescence polarization analysisMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50538812(CHEMBL4635096)
Affinity DataKd:  350nMAssay Description:Binding affinity to CBX6 (unknown origin) assessed as dissociation constant by fluorescence polarization analysisMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50538813(CHEMBL4643012)
Affinity DataKd:  400nMAssay Description:Binding affinity to CBX6 (unknown origin) assessed as dissociation constant by fluorescence polarization analysisMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50538814(CHEMBL4640186)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to CBX6 (unknown origin) assessed as dissociation constant by fluorescence polarization analysisMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50155931(CHEMBL3780251)
Affinity DataKd:  300nMAssay Description:Binding affinity to N-terminal His6-tagged human CBX6 (8 to 65 residues) expressed in Escherichia coli BL21 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50155893(CHEMBL3780712)
Affinity DataKd:  800nMAssay Description:Binding affinity to N-terminal His6-tagged human CBX6 (8 to 65 residues) expressed in Escherichia coli BL21 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50157395(CHEMBL3780663)
Affinity DataKd:  110nMAssay Description:Binding affinity to N-terminal His6-tagged human CBX6 (8 to 65 residues) expressed in Escherichia coli BL21 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50155932(CHEMBL3780489)
Affinity DataKd:  900nMAssay Description:Binding affinity to N-terminal His6-tagged human CBX6 (8 to 65 residues) expressed in Escherichia coli BL21 using FITC-peptide-3 as competitive bindi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChromobox protein homolog 6(Homo sapiens (Human))
University Of Victoria

Curated by ChEMBL
LigandPNGBDBM50157400(CHEMBL3781600)
Affinity DataKd:  910nMAssay Description:Binding affinity to N-terminal His6-tagged human CBX6 (8 to 65 residues) expressed in Escherichia coli BL21 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed