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Found 8 Enz. Inhib. hit(s) with Target = 'Cytoplasmic dynein 1 heavy chain 1'
TargetCytoplasmic dynein 1 heavy chain 1(Rattus norvegicus)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50184425(CHEMBL206161 | Purealin)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of MT-stimulated ATPase activity of rat cytoplasmic dynein heavy chain motor domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytoplasmic dynein 1 heavy chain 1(Rattus norvegicus)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50117089(CHEMBL204484 | CHEMBL83995 | N-[2-(2-Amino-3H-imid...)
Affinity DataIC50:  4.20E+4nMAssay Description:Inhibition of MT-stimulated ATPase activity of rat cytoplasmic dynein heavy chain motor domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytoplasmic dynein 1 heavy chain 1(Rattus norvegicus)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50184427(CHEMBL206373 | Lipopurealin A)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of MT-stimulated ATPase activity of rat cytoplasmic dynein heavy chain motor domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytoplasmic dynein 1 heavy chain 1(Rattus norvegicus)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50184424(3-[2-(3-aminopropoxy)-3,5-dichlorophenyl]-2-hydrox...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of MT-stimulated ATPase activity of rat cytoplasmic dynein heavy chain motor domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytoplasmic dynein 1 heavy chain 1(Rattus norvegicus)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50184426(3-[4-(3-aminopropoxy)-3-bromophenyl]-N-[2-(4-chlor...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of MT-stimulated ATPase activity of rat cytoplasmic dynein heavy chain motor domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytoplasmic dynein 1 heavy chain 1(Rattus norvegicus)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50184421(3-[4-(3-aminopropoxy)-3-bromophenyl]-2-hydroxyimin...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of MT-stimulated ATPase activity of rat cytoplasmic dynein heavy chain motor domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytoplasmic dynein 1 heavy chain 1(Rattus norvegicus)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50184420(3-[2-(3-aminopropoxy)-3,5-dibromophenyl]-2-hydroxy...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of MT-stimulated ATPase activity of rat cytoplasmic dynein heavy chain motor domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytoplasmic dynein 1 heavy chain 1(Rattus norvegicus)
University Of Pittsburgh

Curated by ChEMBL
LigandPNGBDBM50184423(3-[2-(3-aminopropoxy)-3,5-dibromophenyl]-N-[2-(4-c...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of MT-stimulated ATPase activity of rat cytoplasmic dynein heavy chain motor domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed