Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) with Target = 'N-acetyltransferase domain-containing protein'
TargetN-acetyltransferase domain-containing protein(Pseudomonas aeruginosa)
University Of Virginia

LigandPNGBDBM213237(4-Methylumbelliferyl phosphate)
Affinity DataKd:  1.65E+5nMpH: 7.5 T: 2°CAssay Description:Isothermal titration calorimetry (ITC) measurements were performed at 25 °C using an iTC200 calorimeter (MicroCal). Preparations of purified pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-acetyltransferase domain-containing protein(Pseudomonas aeruginosa)
University Of Virginia

LigandPNGBDBM50335523((6R,7R)-3-(acetoxymethyl)-7-(2-(2-aminothiazol-4-y...)
Affinity DataKd:  3.50E+3nMpH: 7.5 T: 2°CAssay Description:Isothermal titration calorimetry (ITC) measurements were performed at 25 °C using an iTC200 calorimeter (MicroCal). Preparations of purified pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-acetyltransferase domain-containing protein(Pseudomonas aeruginosa)
University Of Virginia

LigandPNGBDBM50335563((6R,7R)-3-(carbamoyloxymethyl)-7-methoxy-8-oxo-7-(...)
Affinity DataKd:  4.93E+4nMpH: 7.5 T: 2°CAssay Description:Isothermal titration calorimetry (ITC) measurements were performed at 25 °C using an iTC200 calorimeter (MicroCal). Preparations of purified pr...More data for this Ligand-Target Pair
TargetN-acetyltransferase domain-containing protein(Pseudomonas aeruginosa)
University Of Virginia

LigandPNGBDBM213239(CoA)
Affinity DataKd:  3.90E+3nMpH: 7.5 T: 2°CAssay Description:Isothermal titration calorimetry (ITC) measurements were performed at 25 °C using an iTC200 calorimeter (MicroCal). Preparations of purified pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-acetyltransferase domain-containing protein(Pseudomonas aeruginosa)
University Of Virginia

LigandPNGBDBM50350472(640/359 | Anaptivan | CEFUROXIME | Ceftin)
Affinity DataKd:  1.77E+5nMpH: 7.5 T: 2°CAssay Description:Isothermal titration calorimetry (ITC) measurements were performed at 25 °C using an iTC200 calorimeter (MicroCal). Preparations of purified pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-acetyltransferase domain-containing protein(Pseudomonas aeruginosa)
University Of Virginia

LigandPNGBDBM213238(AcCoA)
Affinity DataKd:  3.80E+3nMpH: 7.5 T: 2°CAssay Description:Isothermal titration calorimetry (ITC) measurements were performed at 25 °C using an iTC200 calorimeter (MicroCal). Preparations of purified pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetN-acetyltransferase domain-containing protein(Pseudomonas aeruginosa)
University Of Virginia

LigandPNGBDBM82898((6R,7R)-3-(acetoxymethyl)-8-keto-7-[[2-(2-thienyl)...)
Affinity DataKd:  1.69E+4nMpH: 7.5 T: 2°CAssay Description:Isothermal titration calorimetry (ITC) measurements were performed at 25 °C using an iTC200 calorimeter (MicroCal). Preparations of purified pr...More data for this Ligand-Target Pair